SCHEMBL3609610

SCHEMBL3609610

CC(C)[C@H](NS(=O)(=O)c1ccc(-c2ccc(NC(=O)c3cc(-c4ccc(Cl)cc4)no3)cc2)cc1)C(=O)O

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 13/20 0.66
MMP13 P45452 6/20 0.63
MMP7 P09237 2/20 0.63
MMP9 P14780 2/20 0.63
MMP1 P03956 1/20 0.63
MMP3 P08254 1/20 0.63
ADAMTS4 O75173 2/20 0.59
MMP12 P39900 2/20 0.59
MMP14 P50281 2/20 0.59
CSGALNACT1 Q8TDX6 4/20 0.57
MMP8 P22894 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3609617 1.00 MMP2 (0.66) MMP2MMP13MMP7MMP9MMP1
SCHEMBL3619101 0.91 MMP2 (0.55) MMP2MMP13MMP7MMP9MMP1
SCHEMBL3619094 0.91 MMP2 (0.55) MMP2MMP13MMP7MMP9MMP1
SCHEMBL3091604 0.82 MMP2 (0.77) MMP2MMP13MMP7MMP9MMP1
SCHEMBL2300240 0.81 CSGALNACT1 (0.84) CSGALNACT1
SCHEMBL2293666 0.81 CSGALNACT1 (0.84) CSGALNACT1
SCHEMBL3618247 0.80 MMP2 (1.00) MMP2MMP13MMP7MMP9MMP1
SCHEMBL7408882 0.79 MMP2 (1.00) MMP2MMP13MMP7MMP9MMP1
SCHEMBL7408889 0.79 MMP2 (1.00) MMP2MMP13MMP7MMP9MMP1
SCHEMBL3612405 0.78 MMP2 (0.64) MMP2MMP13MMP7MMP9MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100137298-A1 Biaryl Sulfonamides and Methods for Using Same WYETH (US) 2010-06-03 US claimed
EP-1692124-B1 BIARYL SULFONAMIDES AS MMP INHIBITORS WYETH CORP (US) 2008-10-15 EP claimed
EP-1692124-A1 BIARYL SULFONAMIDES AS MMP INHIBITORS Wyeth (US) 2006-08-23 EP claimed
WO-2005061477-A1 BIARYL SULFONAMIDES AS MMP INHIBITORS WYETH (US) 2005-07-07 WO claimed
US-20050143422-A1 Biaryl sulfonamides and methods for using same WYETH (US) 2005-06-30 US claimed
US-20100137298-A1 Biaryl Sulfonamides and Methods for Using Same WYETH (US) 2010-06-03 US disclosed
US-20100137298-A1 Biaryl Sulfonamides and Methods for Using Same WYETH (US) 2010-06-03 US disclosed
US-20100137298-A1 Biaryl Sulfonamides and Methods for Using Same WYETH (US) 2010-06-03 US disclosed
EP-1692124-B1 BIARYL SULFONAMIDES AS MMP INHIBITORS WYETH CORP (US) 2008-10-15 EP disclosed
US-7420001-B2 Biaryl sulfonamides and methods for using same WYETH (US) 2008-09-02 US disclosed
US-7420001-B2 Biaryl sulfonamides and methods for using same WYETH (US) 2008-09-02 US disclosed
US-7420001-B2 Biaryl sulfonamides and methods for using same WYETH (US) 2008-09-02 US disclosed
EP-1692124-A1 BIARYL SULFONAMIDES AS MMP INHIBITORS Wyeth (US) 2006-08-23 EP disclosed
WO-2005061477-A1 BIARYL SULFONAMIDES AS MMP INHIBITORS WYETH (US) 2005-07-07 WO disclosed
US-20050143422-A1 Biaryl sulfonamides and methods for using same WYETH (US) 2005-06-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137298-A1 Biaryl Sulfonamides and Methods for Using Same STS, MMP3, AADAC MMP2 5/4885MMP13 13/4885MMP7 35/4885
US-20050143422-A1 Biaryl sulfonamides and methods for using same STS, MMP3, AADAC MMP2 5/4885MMP13 13/4885MMP7 35/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.