SCHEMBL3611539

SCHEMBL3611539

O=C(Cc1csc(N(Cc2cccs2)C(=O)O)n1)NO

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
PDE5A O76074 10/20 0.46
KDM4E B2RXH2 2/20 0.46
PDE1A P54750 4/20 0.45
PDE1B Q01064 4/20 0.45
PDE1C Q14123 4/20 0.45
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
ESR2 Q92731 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPT P10636 3/20 0.41
GAA P10253 1/20 0.41
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3602128 0.83 PDE5A (0.43) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL3609752 0.82 PDE5A (0.43) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL3605700 0.82 NPC1 (0.51) SMN1; SMN2NPC1RAB9AMEN1POLB
SCHEMBL3604375 0.81 PDE5A (0.44) HDAC1HDAC6PDE5AKDM4EPDE1A
SCHEMBL3600139 0.79 GSTO1 (0.52) HDAC1HDAC6PDE5AKDM4EPDE1A
SCHEMBL3603075 0.77 PDE5A (0.45) HDAC1HDAC6SMN1; SMN2RAB9APDE5A
SCHEMBL3600706 0.75 PDE5A (0.43) HDAC1HDAC6PDE5AKDM4EPDE1A
SCHEMBL3615409 0.74 PDE5A (0.42) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL3612348 0.74 PDE5A (0.64) HDAC1HDAC6SMN1; SMN2PDE5AKDM4E
SCHEMBL3602419 0.73 PDE5A (0.46) HDAC1HDAC6PDE5APDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100152188-A1 Novel Heterocyclic Compounds ORCHID RESEARCH LABORATORIES LIMITED (IN) 2010-06-17 US claimed
US-20100152188-A1 Novel Heterocyclic Compounds ORCHID RESEARCH LABORATORIES LIMITED (IN) 2010-06-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100152188-A1 Novel Heterocyclic Compounds CYP11B2, CYP3A5, CYP11B1 HDAC1 307/4885HDAC6 90/4885SMN1; SMN2 3278/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.