SCHEMBL3615280

SCHEMBL3615280

CCOC(=O)c1cnc2ccnn2c1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.49
RAB9A P51151 7/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.48
KDM4E B2RXH2 9/20 0.48
GAA P10253 3/20 0.48
GLA P06280 2/20 0.48
HPGD P15428 6/20 0.47
ALDH1A1 P00352 6/20 0.47
TP53 P04637 3/20 0.47
RXFP1 Q9HBX9 1/20 0.47
HSD17B10 Q99714 2/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
MAPT P10636 2/20 0.44
NFKB1 P19838 2/20 0.44
NFKB2 Q00653 2/20 0.44
RELA Q04206 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3620953 0.85 KDM4E (0.49) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL236467 0.84 RAB9A (0.64) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL6002635 0.82 KDM4E (0.46) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL9678739 0.80 NPC1 (0.47) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL31023504 0.79 KDM4E (0.48) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL6289416 0.78 NPC1 (0.55) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL14471947 0.78 JAK2 (0.47) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL25375133 0.78 CSNK1D (0.49) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL14471980 0.78 P2RY12 (0.44) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL11457347 0.77 KDM4E (0.57) NPC1RAB9ASMN1; SMN2LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119320383-A Nitrogen-containing heteroaryl compound, and preparation method and application thereof 北京鞍石生物科技股份有限公司 2025-01-17 CN disclosed
US-20100069395-A1 Pyrazolo[1,5-a]pyrimidine-3-carboxylic acid compounds as protein kinase inhibitors IMBACH PATRICIA 2010-03-18 US disclosed
EP-2079745-A1 3-AMINOCARBONYI-SUBSTITUTED FUSED PYRAZOLO-DERIVATIVES AS PROTEIN KINASE MODULATORS Novartis AG (CH) 2009-07-22 EP disclosed
WO-2008052964-A1 3-AMINOCARBONYI-SUBSTITUTED FUSED PYRAZOLO-DERIVATIVES AS PROTEIN KINASE MODULATORS NOVARTIS AG (CH) 2008-05-08 WO disclosed
EP-1918291-A1 3-Aminocarbonyl-substituted fused pyrazolo-derivatives as protein kinase modulators Novartis AG (CH) 2008-05-07 EP disclosed
US-3925385-A 6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines VIRATEK, INC., A CORP. OF DE. 1975-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069395-A1 Pyrazolo[1,5-a]pyrimidine-3-carboxylic acid compounds as protein kinase inhibitors PRKCA, PRKACA, MAP3K19 NPC1 2457/4885RAB9A 1142/4885SMN1; SMN2 3346/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.