SCHEMBL361680

SCHEMBL361680

Cc1cc(/C(CC(c2ccc(-c3ccc(C(=O)O)cc3)cc2)c2ccc(Cl)cc2F)=N/O)c[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.47
S1PR3 Q99500 4/20 0.36
S1PR1 P21453 2/20 0.36
BRD4 O60885 1/20 0.33
SRD5A2 P31213 1/20 0.32
MGAM O43451 2/20 0.32
GAA P10253 2/20 0.32
SI P14410 2/20 0.32
MGAM2 Q2M2H8 2/20 0.32
S1PR2 O95136 1/20 0.32
SPR P35270 1/20 0.32
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
ERCC1 P07992 1/20 0.31
ERCC4 Q92889 1/20 0.31
F11 P03951 1/20 0.31
ADRB1 P08588 2/20 0.31
ADRB3 P13945 2/20 0.31
GCGR P47871 1/20 0.31
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363277 0.93 GPBAR1 (0.41) GPBAR1S1PR3S1PR1SRD5A2SPR
SCHEMBL363638 0.93 GPBAR1 (0.41) GPBAR1S1PR3S1PR1SRD5A2SPR
SCHEMBL363248 0.93 GPBAR1 (0.41) GPBAR1S1PR3S1PR1SRD5A2SPR
SCHEMBL363178 0.92 GPBAR1 (0.51) GPBAR1BRD4SRD5A2MGAMGAA
SCHEMBL363089 0.92 GPBAR1 (0.39) GPBAR1S1PR3S1PR1BRD4ERCC1
SCHEMBL364998 0.92 GPBAR1 (0.39) GPBAR1S1PR3S1PR1BRD4ERCC1
SCHEMBL364367 0.92 GPBAR1 (0.39) GPBAR1S1PR3S1PR1BRD4ERCC1
SCHEMBL362281 0.91 GPBAR1 (0.48) GPBAR1BRD4RXRARXRBERCC1
SCHEMBL362457 0.91 GPBAR1 (0.48) GPBAR1BRD4MGAMGAASI
SCHEMBL363327 0.91 GPBAR1 (0.38) GPBAR1S1PR3S1PR1BRD4RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed