SCHEMBL363327

SCHEMBL363327

Cc1cc(/C(CC(c2ccc(-c3ccc(CC(=O)O)cc3)cc2)c2ccc(Cl)cc2F)=N/O)c[nH]c1=O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.38
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
BRD4 O60885 1/20 0.31
DGAT1 O75907 1/20 0.31
PTGS2 P35354 1/20 0.30
FDFT1 P37268 1/20 0.30
MDM2 Q00987 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364696 1.00 GPBAR1 (0.38) GPBAR1S1PR1S1PR3ADRB1ADRB3
SCHEMBL362367 1.00 GPBAR1 (0.38) GPBAR1S1PR1S1PR3ADRB1ADRB3
SCHEMBL361680 0.91 GPBAR1 (0.47) GPBAR1S1PR1S1PR3ADRB1ADRB3
SCHEMBL364367 0.89 GPBAR1 (0.39) GPBAR1S1PR1S1PR3ADRB1ADRB3
SCHEMBL363089 0.89 GPBAR1 (0.39) GPBAR1S1PR1S1PR3ADRB1ADRB3
SCHEMBL364998 0.89 GPBAR1 (0.39) GPBAR1S1PR1S1PR3ADRB1ADRB3
SCHEMBL364313 0.89 S1PR3 (0.36) GPBAR1S1PR1S1PR3
SCHEMBL363638 0.86 GPBAR1 (0.41) GPBAR1S1PR1S1PR3ADRB1ADRB3
SCHEMBL363248 0.86 GPBAR1 (0.41) GPBAR1S1PR1S1PR3ADRB1ADRB3
SCHEMBL363277 0.86 GPBAR1 (0.41) GPBAR1S1PR1S1PR3ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed