SCHEMBL363248

SCHEMBL363248

Cc1cc(C(=O)O)ccc1-c1ccc([C@@H](C/C(=N\O)c2c[nH]c(=O)c(C)c2)c2ccc(Cl)cc2F)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.41
ADRB1 P08588 5/20 0.38
ADRB3 P13945 5/20 0.38
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
RARB P10826 1/20 0.34
SRD5A2 P31213 1/20 0.34
AKR1C3 P42330 2/20 0.33
AKR1C2 P52895 2/20 0.33
TNKS2 Q9H2K2 1/20 0.33
SLC1A3 P43003 1/20 0.32
SLC1A2 P43004 1/20 0.32
SLC1A1 P43005 1/20 0.32
PTGER4 P35408 2/20 0.32
PTGER2 P43116 1/20 0.32
ADH5 P11766 1/20 0.32
SPR P35270 1/20 0.32
EIF4E P06730 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363277 1.00 GPBAR1 (0.41) GPBAR1ADRB1ADRB3S1PR1S1PR3
SCHEMBL363638 1.00 GPBAR1 (0.41) GPBAR1ADRB1ADRB3S1PR1S1PR3
SCHEMBL361680 0.93 GPBAR1 (0.47) GPBAR1ADRB1ADRB3S1PR1S1PR3
SCHEMBL364024 0.92 GPBAR1 (0.42) GPBAR1ADRB1ADRB3RARBSRD5A2
SCHEMBL364066 0.92 GPBAR1 (0.42) GPBAR1ADRB1ADRB3RARBSRD5A2
SCHEMBL363679 0.92 GPBAR1 (0.42) GPBAR1ADRB1ADRB3RARBSRD5A2
SCHEMBL364367 0.87 GPBAR1 (0.39) GPBAR1ADRB1ADRB3S1PR1S1PR3
SCHEMBL364998 0.87 GPBAR1 (0.39) GPBAR1ADRB1ADRB3S1PR1S1PR3
SCHEMBL363089 0.87 GPBAR1 (0.39) GPBAR1ADRB1ADRB3S1PR1S1PR3
SCHEMBL364696 0.86 GPBAR1 (0.38) GPBAR1ADRB1ADRB3S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed