SCHEMBL361815

SCHEMBL361815

C=CCOc1ccccc1C#N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.47
MAPK1 P28482 2/20 0.47
HPGD P15428 2/20 0.47
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 5/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
ADRA2A P08913 2/20 0.45
ADRA2B P18089 2/20 0.45
GAA P10253 2/20 0.45
ADRA2C P18825 1/20 0.45
LIG1 P18858 1/20 0.45
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
HTR1A P08908 1/20 0.42
MAOA P21397 1/20 0.42
HTR2B P41595 1/20 0.42
POLB P06746 1/20 0.42
KDM4E B2RXH2 2/20 0.41
TP53 P04637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2395315 0.86 HPGD (0.43) TSHRMAPK1HPGDHSD17B10ALDH1A1
SCHEMBL3435213 0.84 ADRA2A (0.46) TSHRMAPK1HPGDHSD17B10ALDH1A1
SCHEMBL17329279 0.84 ADRA2A (0.46) TSHRMAPK1HPGDHSD17B10ALDH1A1
SCHEMBL19759485 0.82 ALDH1A1 (0.50) TSHRMAPK1HPGDALDH1A1SMN1; SMN2
SCHEMBL2555115 0.81 ALDH1A1 (0.49) TSHRMAPK1HPGDALDH1A1SMN1; SMN2
SCHEMBL7113700 0.81 LIG1 (0.49) TSHRMAPK1HPGDHSD17B10ALDH1A1
SCHEMBL5134014 0.80 HPGD (0.46) TSHRMAPK1HPGDHSD17B10ALDH1A1
SCHEMBL16112318 0.80 FFAR1 (0.48) TSHRMAPK1HPGDHSD17B10ADRA2A
1,2-Diallyloxybenzene SCHEMBL29768784 0.80 HPGD (0.60) TSHRMAPK1HPGDHSD17B10ALDH1A1
1,2-Diallyloxybenzene SCHEMBL366516 0.80 HPGD (0.60) TSHRMAPK1HPGDHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104311474-B Synthesis method of 3-alkynyl pyridine compound 河南师范大学 2017-01-11 CN disclosed
CN-104311474-A Synthesis method of 3-alkynyl pyridine compound UNIV HENAN NORMAL 2015-01-28 CN disclosed
EP-2593461-A1 COMPOUNDS FOR THE REDUCTION OF BETA-AMYLOID PRODUCTION Bristol-Myers Squibb Company (US) 2013-05-22 EP disclosed
WO-2012009309-A1 COMPOUNDS FOR THE REDUCTION OF BETA-AMYLOID PRODUCTION BRISTOL-MYERS SQUIBB COMPANY (US) 2012-01-19 WO disclosed
US-6008401-A CONDENSATION REACTION BETWEEN 4-HALO OR NITRO SUBSTITUTED BENZONITRILE DERIVATIVE AND OTICALLY ACTIVE ALCOHOL PRODUCES AN OPTICALLY ACTIVE ALKOXYBENZONITRILE DERIVATIVE NIPPON OIL CO., LTD. (JP) 1999-12-28 US disclosed
US-5380654-A Process for the preparation of epoxides of means of microorganisms JAPAN ENERGY CORPORATION (JP) 1995-01-10 US disclosed
US-5376539-A Aerobic incubation of allyl phenyl ether with arthrobacter, brevibacterium, corynebacterium, pseudomonas or rhodococcus yields glycidyl phenyl ether NIPPON MINING CO., LTD. (JP) 1994-12-27 US disclosed
EP-0166527-B1 A PROCESS FOR THE PREPARATION OF EPOXIDES BY MEANS OF MICROORGANISMS NIPPON MINING COMPANY LIMITED (JP) 1991-04-03 EP disclosed
EP-0411787-A2 Microbiological production of 2,3-epoxypropyl ethers IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-02-06 EP disclosed
EP-0166527-A2 A process for the preparation of epoxides by means of microorganisms NIPPON MINING COMPANY LIMITED (JP) 1986-01-02 EP disclosed