Tamibarotene

Tamibarotene

SCHEMBL36207

CC1(C)CCC(C)(C)c2cc(NC(=O)c3ccc(C(=O)O)cc3)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

RARARARB

The experimentally established mechanism targets of Tamibarotene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB known ✓ P10826 10/20 1.00
RARA known ✓ P10276 8/20 1.00
RARG P13631 10/20 1.00
CYP26A1 O43174 5/20 1.00
CYP3A4 P08684 3/20 1.00
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
PGR P06401 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
TBXA2R P21731 1/20 1.00
BLVRB P30043 1/20 1.00
ALDH1A1 P00352 1/20 0.84
CYP1A2 P05177 1/20 0.84
CYP2C9 P11712 1/20 0.84
TSHR P16473 1/20 0.84
MAPK1 P28482 1/20 0.84
CYP2C19 P33261 1/20 0.84
CYP26B1 Q9NR63 2/20 0.74
RXRA P19793 11/20 0.62
RXRB P28702 9/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tamibarotene SCHEMBL29373818 1.00 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
Tamibarotene SCHEMBL21055743 0.99 RARB (0.97) RARBRARGRARACYP26A1CYP3A4
Tamibarotene SCHEMBL21274219 0.92 RARB (0.85) RARBRARGRARACYP26A1CYP3A4
SCHEMBL726740 0.91 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL29355626 0.91 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
Tamibarotene SCHEMBL21274122 0.91 RARB (0.83) RARBRARGRARACYP26A1CYP3A4
SCHEMBL22872722 0.91 RARB (0.83) RARBRARGRARACYP26A1CYP3A4
SCHEMBL17832980 0.91 RARB (0.83) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8461601 0.90 CYP26A1 (0.82) RARBRARGRARACYP26A1CYP3A4
SCHEMBL1615110 0.89 RARA (0.80) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5276 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4745155-A1 POWDER CONTAINING PARTICLES OF GELATIN DERIVATIVE AND APPLICATION OF SAME IN MEDICAL TREATMENT National Institute for Materials Science (JP) 2026-05-20 EP claimed
EP-4744657-A1 THERAPEUTIC AGENT FOR HUMAN GRAFT VERSUS HOST DISEASE AND COMBINATION THEREOF National University Corporation Okayama University (JP) 2026-05-20 EP claimed
US-20260124164-A1 PHARMACEUTICAL COMPOSITION FOR TREATING AUTOSOMAL DOMINANT POLYCYSTIC KIDNEY DISEASE KYOTO UNIVERSITY (JP) 2026-05-07 US claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
US-12589189-B2 Use of retinoic acid receptor (RAR) agonists for reversing, preventing, or delaying calcification of aortic valve INSERM (INSTITUTE NATIONAL DE LA SANTA ET DE LA RECHERCHE MEDICALE) (FR) 2026-03-31 US claimed
EP-4037672-B1 RETINOIC ACID RECEPTOR (RAR) AGONISTS FOR REVERSING, PREVENTING, OR DELAYING CALCIFICATION OF AORTIC VALVE INST NAT SANTE RECH MED (FR) 2026-03-11 EP claimed
US-12548678-B2 Methods and systems for machine learning analysis of single nucleotide polymorphisms in lupus AMPEL BIOSOLUTIONS, LLC (US) 2026-02-10 US claimed
US-12521358-B2 Method for selecting cancer patients for whom combination therapy with retinoid and cancer therapeutic agent is effective, and combination medicament with retinoid and cancer therapeutic agent RAQUALIA PHARMA INC. (JP) 2026-01-13 US claimed
US-12514834-B2 Pharmaceutical composition for treating and/or preventing renal cystic ciliopathy KYOTO UNIVERSITY (JP) 2026-01-06 US claimed
US-20260000697-A1 COMBINATION FORMULATION OF CEDAZURIDINE OTSUKA PHARMA CO LTD (JP) 2026-01-01 US claimed
EP-0478787-B1 NOVEL PROCESS FOR PRODUCING BENZOIC ACID DERIVATIVE SHIONOGI & CO (JP) 1994-12-21 EP claimed
EP-0625045-A1 METHODS OF TREATING INFLAMMATORY DERMATOSES Kligman, Albert M. (US) 1994-11-23 EP claimed
EP-0619116-A2 Use of synthetic retinoids for osteopathy HOECHST JAPAN LIMITED (JP) 1994-10-12 EP claimed
EP-0465343-B1 Pharmaceutical or cosmetical composition comprising a retinoid and a sterol in association CIRD GALDERMA (FR) 1994-06-15 EP claimed
WO-1993015740-A1 METHODS OF TREATING INFLAMMATORY DERMATOSES KLIGMAN ALBERT M (US) 1993-08-19 WO claimed
US-5214202-A Retinoid activity SHIONOGI & CO., LTD. (JP) 1993-05-25 US claimed
EP-0478787-A1 NOVEL PROCESS FOR PRODUCING BENZOIC ACID DERIVATIVE SHIONOGI & CO., LTD. (JP) 1992-04-08 EP claimed
EP-0170105-B1 BENZOIC ACID DERIVATIVES Shudo, Koichi, Prof. Dr. (JP) 1990-10-17 EP claimed
US-4703110-A Benzoic acid derivatives having a para substituent which is a substituted phenyl group connected by a linking radical; useful in neoplastic cell differentiation and diagnosis Shudo, Koichi (JP) 1987-10-27 US claimed
EP-0170105-A2 Benzoic acid derivatives Shudo, Koichi, Prof. Dr. (JP) 1986-02-05 EP claimed