SCHEMBL3622982

SCHEMBL3622982

FC(F)(F)c1ncc2ccccc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
GAA P10253 2/20 0.43
ALDH1A1 P00352 2/20 0.43
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GPR3 P46089 1/20 0.42
EGFR P00533 1/20 0.42
CCNE2 O96020 3/20 0.41
CCNE1 P24864 3/20 0.41
CDK2 P24941 3/20 0.41
MEN1 O00255 2/20 0.41
POLB P06746 2/20 0.41
KMT2A Q03164 2/20 0.41
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
NPC1 O15118 1/20 0.41
THRB P10828 1/20 0.41
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TLR7 Q9NYK1 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30200294 1.00 MAPT (0.43) MAPTGAAALDH1A1RAB9AKDM4E
Biphenyl SCHEMBL27928291 0.93 GAA (0.42) MAPTGAAALDH1A1RAB9AKDM4E
SCHEMBL30562839 0.84 KDM4E (0.39) MAPTGAAALDH1A1RAB9AKDM4E
SCHEMBL19032530 0.82 KDM4E (0.38) MAPTGAAALDH1A1RAB9AKDM4E
SCHEMBL10704355 0.81 KDM4E (0.43) MAPTALDH1A1KDM4EGPR3EGFR
SCHEMBL10707622 0.81 KDM4E (0.43) MAPTALDH1A1KDM4EGPR3EGFR
SCHEMBL322264 0.79 CYP1A2 (0.42) MAPTALDH1A1KDM4EGPR3EGFR
SCHEMBL31391354 0.76 ALDH1A1 (0.43) MAPTGAAALDH1A1RAB9AKDM4E
SCHEMBL30071208 0.76 MALT1 (0.49) MAPTGAAALDH1A1RAB9AKDM4E
SCHEMBL30368951 0.76 CYP1A2 (0.40) MAPTGAAALDH1A1KDM4EGPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106414430-A Pharmacologically active quinazolinedione derivatives 奥赖恩公司 2017-02-15 CN claimed
CN-103910688-A 2-propyl-4-chloroquinazoline derivative, its preparation method thereof and its application thereof CHUNLIN CHEN 2014-07-09 CN claimed
CN-101679311-A Quinazoline compound WYETH CORP 2010-03-24 CN claimed
EP-2142517-A2 QUINAZOLINE COMPOUNDS Wyeth (US) 2010-01-13 EP claimed
WO-2009020683-A2 QUINAZOLINE COMPOUNDS WYETH (US) 2009-02-12 WO claimed
WO-2025022007-A1 PESTICIDALLY ACTIVE QUINAZOLINE COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2025-01-30 WO disclosed
CN-117561252-A 2- [3- [1[ (quinazolin-4-yl) amino ] ethyl ] pyrazin-2-yl ] thiazole-5-carbonitrile derivatives and similar compounds as pesticides 先正达农作物保护股份公司 2024-02-13 CN disclosed
WO-2024030647-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS THERAS, INC. (US) 2024-02-08 WO disclosed
US-20240032541-A1 HERBICIDAL COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2024-02-01 US disclosed
WO-2024008179-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE, LTD. (KY) 2024-01-11 WO disclosed
CN-114436975-B 2-trifluoromethyl-4-aminoquinazoline compound and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2023-10-31 CN disclosed
WO-2023179703-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-09-28 WO disclosed
EP-0545491-B1 Photographic silver halide colour materials KODAK LTD (GB) 1998-10-14 EP disclosed
EP-0565165-B1 Photographic silver halide colour materials KODAK LTD (GB) 1998-09-02 EP disclosed
EP-0760819-A1 TRICYCLIC DICARBONYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed
WO-1995032205-A1 TRICYCLIC DICARBONYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1995-11-30 WO disclosed
US-5415981-A Sulfohydrazide developer, heteroarylacetonitrile color coupler EASTMAN KODAK COMPANY (US) 1995-05-16 US disclosed
US-5284739-A Devloper and coupler present in drops of a high-boiling solvent; water pollution control EASTMAN KODAK COMPANY (US) 1994-02-08 US disclosed
EP-0565165-A1 Photographic silver halide colour materials KODAK LIMITED (GB) 1993-10-13 EP disclosed
EP-0545491-A1 Photographic silver halide colour materials KODAK LIMITED (GB) 1993-06-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240032541-A1 HERBICIDAL COMPOUNDS HAX1, DDT, MTX1 MAPT 4243/4885GAA 604/4885ALDH1A1 264/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.