SCHEMBL3625089

SCHEMBL3625089

CC(C)(Cc1cccc(CC(=O)NCc2ccccc2)c1)NC[C@H](O[Si](C)(C)C(C)(C)C)c1ccc(O)c(NC=O)c1

nearest known ligand 0.59

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 20/20 0.59
CHRM3 P20309 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3625091 1.00 ADRB2 (0.59) ADRB2CHRM3
SCHEMBL3627176 0.92 ADRB2 (0.50) ADRB2CHRM3
SCHEMBL3627170 0.92 ADRB2 (0.50) ADRB2CHRM3
SCHEMBL3629058 0.91 ADRB2 (0.46) ADRB2
SCHEMBL3629054 0.91 ADRB2 (0.46) ADRB2
SCHEMBL13807627 0.89 ADRB2 (0.44) ADRB2
SCHEMBL5069535 0.89 ADRB2 (0.63) ADRB2CHRM3
SCHEMBL5580669 0.89 ADRB2 (0.63) ADRB2CHRM3
SCHEMBL3619535 0.86 ADRB2 (0.45) ADRB2
SCHEMBL3619529 0.86 ADRB2 (0.45) ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796283-B2 Indole and azaindole modulators of the alpha 7 nachr PROXIMAGEN LIMITED (GB) 2014-08-05 US disclosed
EP-1730103-B1 FORMAMIDE DERIVATIVES USEFUL AS ADRENOCEPTOR PFIZER LTD (GB) 2010-05-26 EP disclosed
US-7547731-B2 Formamide derivatives for the treatment of diseases PFIZER INC (US) 2009-06-16 US disclosed
US-7547731-B2 Formamide derivatives for the treatment of diseases PFIZER INC (US) 2009-06-16 US disclosed
US-20080207689-A1 Formamide Derivatives For The Treatment of Diseases PFIZER INC 2008-08-28 US disclosed
US-20080207689-A1 Formamide Derivatives For The Treatment of Diseases PFIZER INC 2008-08-28 US disclosed
US-7241810-B2 Formamide derivatives for the treatment of diseases PFIZER INC (US) 2007-07-10 US disclosed
US-7241810-B2 Formamide derivatives for the treatment of diseases PFIZER INC (US) 2007-07-10 US disclosed
US-20050215590-A1 Formamide derivatives for the treatment of diseases PFIZER LIMITED (GB) 2005-09-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080207689-A1 Formamide Derivatives For The Treatment of Diseases FH, FAH, HRH4 ADRB2 751/4885CHRM3 927/4885
US-20050215590-A1 Formamide derivatives for the treatment of diseases FH, FAH, HRH4 ADRB2 751/4885CHRM3 927/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.