SCHEMBL362689

SCHEMBL362689

COC(=O)c1ccc(-c2ccc(C(CC(=O)c3c[nH]c(=O)c(C)c3)c3ccccc3C)cc2)cc1F

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.38
ACLY P53396 1/20 0.38
BRD4 O60885 1/20 0.37
NR4A2 P43354 1/20 0.37
GPBAR1 Q8TDU6 2/20 0.37
MGAM O43451 5/20 0.36
GAA P10253 5/20 0.36
SI P14410 5/20 0.36
MGAM2 Q2M2H8 5/20 0.36
NPC1 O15118 1/20 0.35
CTSA P10619 3/20 0.35
FFAR1 O14842 2/20 0.35
ALDH1A1 P00352 2/20 0.35
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363538 0.85 TDP1 (0.38) TDP1ACLYBRD4MGAMGAA
SCHEMBL364504 0.83 GPBAR1 (0.40) ACLYBRD4NR4A2GPBAR1NPC1
SCHEMBL363216 0.82 GPBAR1 (0.39) ACLYBRD4NR4A2GPBAR1NPC1
SCHEMBL14894610 0.82 GPBAR1 (0.52) TDP1BRD4GPBAR1MGAMGAA
SCHEMBL1390186 0.82 GPBAR1 (0.38) TDP1BRD4NR4A2GPBAR1CTSA
SCHEMBL369861 0.82 GPBAR1 (0.55) TDP1GPBAR1CTSAFFAR1S1PR1
SCHEMBL362317 0.81 GPBAR1 (0.52) BRD4GPBAR1CTSAFFAR1S1PR1
SCHEMBL14896301 0.81 BRD4 (0.48) TDP1BRD4GPBAR1MGAMGAA
SCHEMBL363934 0.79 GPBAR1 (0.47) TDP1BRD4GPBAR1MGAMGAA
SCHEMBL364664 0.78 GAA (0.42) BRD4GPBAR1MGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed