SCHEMBL363216

SCHEMBL363216

COC(=O)c1ccc(-c2ccc(C(C/C(=N\O)c3c[nH]c(=O)c(C)c3)c3ccccc3C)c(F)c2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.39
ACLY P53396 1/20 0.35
NPC1 O15118 1/20 0.34
CTSA P10619 8/20 0.34
FFAR1 O14842 1/20 0.34
NR4A2 P43354 1/20 0.33
ROCK2 O75116 2/20 0.33
ROCK1 Q13464 2/20 0.33
BRD4 O60885 1/20 0.33
CYP3A4 P08684 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363245 0.92 GPBAR1 (0.43) GPBAR1CTSAFFAR1BRD4CYP3A4
SCHEMBL361842 0.87 GPBAR1 (0.51) GPBAR1CTSAFFAR1BRD4CYP3A4
SCHEMBL364504 0.86 GPBAR1 (0.40) GPBAR1ACLYNPC1CTSAFFAR1
SCHEMBL363831 0.85 GPBAR1 (0.42) GPBAR1CTSABRD4
SCHEMBL363688 0.84 GPBAR1 (0.38) GPBAR1CTSABRD4CYP3A4
SCHEMBL362317 0.84 GPBAR1 (0.52) GPBAR1CTSAFFAR1BRD4CYP3A4
SCHEMBL1389910 0.83 GPBAR1 (0.40) GPBAR1NPC1CTSAFFAR1NR4A2
SCHEMBL1389912 0.83 GPBAR1 (0.40) GPBAR1NPC1CTSAFFAR1NR4A2
SCHEMBL362689 0.82 TDP1 (0.38) GPBAR1ACLYNPC1CTSAFFAR1
SCHEMBL362892 0.81 GPBAR1 (0.39) GPBAR1CTSAFFAR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed