SCHEMBL364504

SCHEMBL364504

COC(=O)c1ccc(-c2ccc(C(C/C(=N\O)c3c[nH]c(=O)c(C)c3)c3ccccc3Cl)cc2)cc1F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.40
ACLY P53396 2/20 0.38
CTSA P10619 8/20 0.35
BRD4 O60885 1/20 0.34
NR4A2 P43354 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
FFAR1 O14842 1/20 0.33
NPC1 O15118 1/20 0.33
F9 P00740 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL361844 0.92 GPBAR1 (0.44) GPBAR1ACLYCTSABRD4FFAR1
SCHEMBL363216 0.86 GPBAR1 (0.39) GPBAR1ACLYCTSABRD4NR4A2
SCHEMBL362317 0.85 GPBAR1 (0.52) GPBAR1CTSABRD4FFAR1
SCHEMBL362527 0.84 GPBAR1 (0.55) GPBAR1CTSABRD4MEN1KMT2A
SCHEMBL363538 0.84 TDP1 (0.38) ACLYCTSABRD4PDE3BPDE3A
SCHEMBL363787 0.83 GPBAR1 (0.38) GPBAR1BRD4FFAR1F9
SCHEMBL362646 0.83 GPBAR1 (0.38) GPBAR1BRD4FFAR1F9
SCHEMBL363296 0.83 GPBAR1 (0.38) GPBAR1BRD4FFAR1F9
SCHEMBL364524 0.83 PTGS2 (0.36) GPBAR1CTSABRD4NPC1F9
SCHEMBL362689 0.83 TDP1 (0.38) GPBAR1ACLYCTSABRD4NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed