SCHEMBL362820

SCHEMBL362820

Nc1ccc(Oc2ccc(N)cc2N)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.57
ALDH1A1 P00352 7/20 0.57
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
CYP1A2 P05177 2/20 0.57
CYP2C9 P11712 2/20 0.57
CYP2C19 P33261 2/20 0.57
KDM4E B2RXH2 2/20 0.57
CYP2D6 P10635 1/20 0.57
HPGD P15428 1/20 0.57
CYP3A4 P08684 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
TSHR P16473 1/20 0.56
GAA P10253 2/20 0.50
MITF O75030 1/20 0.50
GFER P55789 1/20 0.50
NLRP1 Q9C000 1/20 0.50
NOD2 Q9HC29 1/20 0.50
MAOA P21397 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30744926 1.00 MAPT (0.57) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7806773 0.98 MAPT (0.59) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL11287510 0.93 ALDH1A1 (0.61) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL28806097 0.91 MAPT (0.53) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL27741074 0.91 MAPT (0.53) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL20347022 0.88 MAPT (0.48) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7024360 0.88 ALDH1A1 (0.50) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL13783383 0.88 TEAD4 (0.61) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL11523227 0.88 MAPT (0.76) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL3193820 0.88 MAPT (0.50) MAPTALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 297 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024100569-A1 SUNSCREEN FORMULATION COMPRISING MICROCAPSULES, AND PROCESS FOR MANUFACTURING SUCH MICROCAPSULES COSMETIC DEVELOPMENT GROUP (FR) 2024-05-16 WO claimed
US-20230292753-A1 AN INSECTICIDAL COMPOSITION FOR PEST CONTROL COMPRISING OF DIACYLHYDRAZINES RAJDHANI PETROCHEMICALS PRIVATE LIMITED (IN) 2023-09-21 US claimed
US-20230284619-A1 Agrochemical mixtures of diamides, plant health additives and insecticide RAJDHANI PETROCHEMICALS PRIVATE LIMITED (IN) 2023-09-14 US claimed
EP-2349551-B2 BENEFIT AGENT CONTAINING DELIVERY PARTICLE PROCTER & GAMBLE (US) 2023-07-26 EP claimed
WO-2022258476-A1 ENCAPSULATED QUATERNARY AMMONIUM COMPOUNDS AND PROCESS FOR PREPARATION THEREOF CLARIANT INTERNATIONAL LTD (CH) 2022-12-15 WO claimed
CN-114805805-A Polyimide with high bonding strength and preparation method and application thereof 中国科学院深圳先进技术研究院 2022-07-29 CN claimed
WO-2022009224-A1 AN INSECTICIDAL COMPOSITION FOR PEST CONTROL COMPRISING OF DIACYLHYDRAZINES RAJDHANI PETROCHEMICALS PRIVATE LIMITED (IN) 2022-01-13 WO claimed
US-11059015-B2 Microcapsules modified with nanomaterial for controlled release of active agent and process for preparation thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2021-07-13 US claimed
EP-3307428-B1 PROCESS FOR THE PREPARATION OF MICROCAPSULES MODIFIED WITH NANOMATERIAL FOR CONTROLLED RELEASE OF ACTIVE AGENT COUNCIL SCIENT IND RES (IN) 2021-01-20 EP claimed
EP-3217793-B1 MICROCAPSULE COMPOSITION CONTAINING WATERSOLUBLE AMINE AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL SCIENT IND RES (IN) 2020-09-09 EP claimed
US-5698731-A REACTING ALKYL CARBONATE AND AROMATIC AMINES IN PRESENCE OF CARBAMATION CATALYST SELECTED FROM N,N-DISUBSTITUTED CARBAMATE COMPLEXS OF ZINC OR COPPER Ministero Dell `Universita` e Della Ricerca Scientifica e Tecnologica (IT) 1997-12-16 US claimed
US-5688988-A REACTION OF AN ORGANIC CARBONATE WITH AROMATIC AMINE USING A ZINC AND/OR COPPER CARBONATE HYDROXIDE CATALYST MINISTERO DELL'UNIVERSITA' E DELLA RICERCA SCIENTIFICA E TECHNOLOGICA (IT) 1997-11-18 US claimed
EP-0752414-A1 Process for the production of aromatic urethanes MINISTERO DELL' UNIVERSITA' E DELLA RICERCA SCIENTIFICA E TECNOLOGICA (IT) 1997-01-08 EP claimed
EP-0752413-A1 Process for the production of aromatic carbamates MINISTERO DELL' UNIVERSITA' E DELLA RICERCA SCIENTIFICA E TECNOLOGICA (IT) 1997-01-08 EP claimed
EP-0214936-B1 PROCESS FOR PRODUCING MICROCAPSULES CIBA-GEIGY AG (CH) 1992-07-08 EP claimed
US-4938797-A Process for the preparation of microcapsules CIBA-GEIGY CORPORATION (US) 1990-07-03 US claimed
EP-0214936-A2 Process for producing microcapsules CIBA-GEIGY AG (CH) 1987-03-18 EP claimed
US-4390596-A POLYAMINE, BIS-MALEIMIDE, FREE RADICAL CATALYST, FILLER RHONE-POULENC INDUSTRIES (FR) 1983-06-28 US claimed
US-4238591-A BIS-MALEIMIDE, SILANEDIOL OR SILOXANE RHONE-POULENC INDUSTRIES (FR) 1980-12-09 US claimed
US-4225498-A Preparation of N-substituted oligo-imides RHONE-POULENC INDUSTRIES (FR) 1980-09-30 US claimed