SCHEMBL362830

SCHEMBL362830

C/C(=N/O)[C@](c1ccc(C2CCNCC2)cc1)(c1ccnc(C)c1)c1ccccc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 9/20 0.38
TLR7 Q9NYK1 9/20 0.38
TLR8 Q9NR97 8/20 0.37
HTR2C P28335 6/20 0.35
SIGMAR1 Q99720 3/20 0.33
SLC18A3 Q16572 1/20 0.33
HTR1A P08908 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
ADRB3 P13945 2/20 0.33
ADRA2B P18089 2/20 0.33
DRD1 P21728 2/20 0.33
DRD5 P21918 2/20 0.33
ADRA1B P35368 2/20 0.33
P2RY14 Q15391 2/20 0.33
TMEM97 Q5BJF2 2/20 0.33
BMPR1B O00238 1/20 0.32
BMPR1A P36894 1/20 0.32
ACVR1B P36896 1/20 0.32
ACVRL1 P37023 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364452 0.90 GPBAR1 (0.31)
SCHEMBL363321 0.88 TLR9 (0.36) TLR9TLR7TLR8HTR2CHTR1A
SCHEMBL362899 0.84 TLR8 (0.40) TLR9TLR7TLR8
SCHEMBL364180 0.82 GPBAR1 (0.35)
SCHEMBL364963 0.81 GPBAR1 (0.32) TLR7TLR8
SCHEMBL363805 0.81 GPBAR1 (0.31)
SCHEMBL364263 0.81 GPBAR1 (0.31)
SCHEMBL364539 0.80 POLB (0.32)
SCHEMBL364836 0.80 POLB (0.32)
SCHEMBL364583 0.79 TLR9 (0.38) TLR9TLR7TLR8HTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed