SCHEMBL364583

SCHEMBL364583

Cc1cc([C@@](C/C=N/O)(c2ccc(C3CCNCC3)cc2)c2ccccc2C)ccn1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 10/20 0.38
TLR7 Q9NYK1 10/20 0.38
TLR8 Q9NR97 9/20 0.38
HTR2C P28335 5/20 0.34
HTR1A P08908 2/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC18A3 Q16572 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
SLC6A3 Q01959 1/20 0.32
NMT1 P30419 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364225 0.84 TLR8 (0.39) TLR9TLR7TLR8GPBAR1
SCHEMBL362361 0.84 GPBAR1 (0.31) GPBAR1
SCHEMBL371360 0.84 PROKR1 (0.38) TLR9TLR7TLR8GPBAR1
SCHEMBL363962 0.82
SCHEMBL364581 0.82
SCHEMBL364230 0.81
SCHEMBL362561 0.80 RAB9A (0.32)
SCHEMBL362830 0.79 TLR9 (0.38) TLR9TLR7TLR8HTR2CHTR1A
SCHEMBL364312 0.79 SMO (0.33)
SCHEMBL363555 0.78 ACSS2 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed