SCHEMBL3628372

SCHEMBL3628372

COc1nc(NC2CCC(NC(=O)O)CC2)c(F)cc1C#N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.53
ROCK1 Q13464 1/20 0.53
GAA P10253 2/20 0.47
PDE4A P27815 3/20 0.38
PDE4B Q07343 3/20 0.38
PDE4C Q08493 3/20 0.38
PDE4D Q08499 3/20 0.38
HPGD P15428 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
IRAK4 Q9NWZ3 3/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
KDM1A O60341 1/20 0.36
NSD2 O96028 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3628370 1.00 ROCK2 (0.53) ROCK2ROCK1GAAPDE4APDE4B
SCHEMBL3627682 0.89 GAA (0.49) ROCK2ROCK1GAAPDE4APDE4B
SCHEMBL3627678 0.89 GAA (0.49) ROCK2ROCK1GAAPDE4APDE4B
SCHEMBL3627803 0.88 LMNA (0.49) ROCK2ROCK1GAAPDE4APDE4B
SCHEMBL3628130 0.88 ROCK2 (0.43) ROCK2ROCK1GAAPDE4APDE4B
SCHEMBL3627799 0.88 LMNA (0.49) ROCK2ROCK1GAAPDE4APDE4B
SCHEMBL3628132 0.88 ROCK2 (0.43) ROCK2ROCK1GAAPDE4APDE4B
SCHEMBL3630214 0.87 GAA (0.47) ROCK2ROCK1GAAHPGDRXFP1
SCHEMBL3630218 0.87 GAA (0.47) ROCK2ROCK1GAAHPGDRXFP1
SCHEMBL3630694 0.86 ROCK2 (0.41) ROCK2ROCK1PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010032875-A2 HETEROCYCLIC CARBOXAMIDE COMPOUNDS ASTELLAS PHARMA INC. (JP) 2010-03-25 WO disclosed