SCHEMBL363023

SCHEMBL363023

Cc1cc(C)c(C=O)c(C)c1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.44
MAPT P10636 3/20 0.44
ERN1 O75460 4/20 0.41
SRC P12931 3/20 0.39
IGF1R P08069 2/20 0.39
AXL P30530 2/20 0.39
PTK2 Q05397 2/20 0.39
AURKB Q96GD4 2/20 0.39
ALK Q9UM73 2/20 0.39
HDAC3 O15379 1/20 0.39
NUAK1 O60285 1/20 0.39
MET P08581 1/20 0.39
PIM1 P11309 1/20 0.39
AKT1 P31749 1/20 0.39
KDR P35968 1/20 0.39
NEK2 P51955 1/20 0.39
PLK1 P53350 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
PKN1 Q16512 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29516419 1.00 CYP3A4 (0.44) CYP3A4MAPTERN1SRCIGF1R
SCHEMBL25342989 0.83 CYP3A4 (0.48) CYP3A4MAPTERN1USP2ALB
SCHEMBL6551606 0.83 CYP3A4 (0.38) CYP3A4MAPTERN1SRCUSP2
SCHEMBL204976 0.82 CYP3A4 (0.44) CYP3A4MAPTERN1SRCIGF1R
SCHEMBL23791666 0.81 ERN1 (0.42) CYP3A4MAPTERN1SRCIGF1R
SCHEMBL1313257 0.78 CYP3A4 (0.35) CYP3A4MAPTERN1USP2ALB
SCHEMBL22379887 0.78 CYP1A2 (0.46) CYP3A4MAPTSRCUSP2CA1
SCHEMBL3269164 0.77 CYP3A4 (0.48) CYP3A4MAPTERN1USP2ALB
SCHEMBL19400788 0.76 CA1 (0.37) CYP3A4MAPTSRCCA1CA2
SCHEMBL17311322 0.76 CYP3A4 (0.52) CYP3A4MAPTERN1USP2ALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 124 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250059349-A1 ELASTOMER COMPOSITION BASED ON AT LEAST ONE NITRILE OXIDE COMPOUND COMPRISING AN EPOXY GROUP COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2025-02-20 US disclosed
EP-4453041-A1 POLYMER CARRYING SPECIFIC EPOXY FUNCTIONAL PENDANT GROUPS COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2024-10-30 EP disclosed
EP-4452957-A1 1,3-DIPOLAR COMPOUND COMPRISING AN EPOXY GROUP AND ITS SYNTHESIS INTERMEDIATES COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2024-10-30 EP disclosed
EP-4453042-A1 ELASTOMER COMPOSITION BASED ON AT LEAST ONE NITRILE OXIDE COMPOUND COMPRISING AN EPOXY GROUP COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2024-10-30 EP disclosed
US-12091540-B2 Grafted polymer bearing pendent cyclic carbonate functional groups COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2024-09-17 US disclosed
US-11952438-B2 1,3-dipolar compound comprising an epoxide group COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2024-04-09 US disclosed
EP-3145909-B1 1,3-DIPOLAR COMPOUND COMPRISING AN ESTER FUNCTION OF CARBOXYLIC ACID AND RUBBER COMPOSITION CONTAINING SAME MICHELIN & CIE (FR) 2023-11-01 EP disclosed
EP-3145909-B1 1,3-DIPOLAR COMPOUND COMPRISING AN ESTER FUNCTION OF CARBOXYLIC ACID AND RUBBER COMPOSITION CONTAINING SAME MICHELIN & CIE (FR) 2023-11-01 EP disclosed
WO-2023117844-A1 1,3-DIPOLAR COMPOUND COMPRISING AN EPOXY GROUP AND ITS SYNTHESIS INTERMEDIATES COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2023-06-29 WO disclosed
WO-2023117840-A1 POLYMER CARRYING SPECIFIC EPOXY FUNCTIONAL PENDANT GROUPS COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2023-06-29 WO disclosed
US-20130123418-A1 RUBBER COMPOSITION CONTAINING A MODIFED ELASTOMER, METHOD FOR PREPARING SAME, AND TIRE CONTAINING SAME MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2013-05-16 US disclosed
US-20130123418-A1 RUBBER COMPOSITION CONTAINING A MODIFED ELASTOMER, METHOD FOR PREPARING SAME, AND TIRE CONTAINING SAME MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2013-05-16 US disclosed
WO-2012007442-A1 RUBBER COMPOSITION CONTAINING A MODIFIED ELASTOMER, METHOD FOR PREPARING SAME, AND TIRE CONTAINING SAME SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2012-01-19 WO disclosed
WO-2012007442-A1 RUBBER COMPOSITION CONTAINING A MODIFIED ELASTOMER, METHOD FOR PREPARING SAME, AND TIRE CONTAINING SAME SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2012-01-19 WO disclosed
WO-2012007441-A1 GRAFT POLYMER TO WHICH COMBINED NITROGEN MOLECULES ARE GRAFTED SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2012-01-19 WO disclosed
WO-2012007441-A1 GRAFT POLYMER TO WHICH COMBINED NITROGEN MOLECULES ARE GRAFTED SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2012-01-19 WO disclosed
WO-2012007684-A1 MOLECULES HAVING COMBINABLE GROUPS ARKEMA FRANCE (FR) 2012-01-19 WO disclosed
EP-0212095-B1 THERMOSETTABLE COMPOUNDS PREPARED FROM MONOHYDROXY AROMATIC ALDEHYDES AND METHYLATED PYRIDINES OR PYRAZINES THE DOW CHEMICAL COMPANY (US) 1989-09-06 EP disclosed
EP-0212095-A1 Thermosettable compounds prepared from monohydroxy aromatic aldehydes and methylated pyridines or pyrazines THE DOW CHEMICAL COMPANY (US) 1987-03-04 EP disclosed
US-4600767-A Thermostable hydroxystyrylaza compounds THE DOW CHEMICAL COMPANY (US) 1986-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11952438-B2 1,3-dipolar compound comprising an epoxide group DCLRE1A, ECH1, ERCC1 CYP3A4 1526/4885MAPT 3139/4885ERN1 152/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.