SCHEMBL3631359

SCHEMBL3631359

Cc1c(C(=O)O)c2cc(=O)ccc-2cn1-c1ccccc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
TP53 P04637 2/20 0.38
HSP90AA1 P07900 2/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
POLB P06746 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
DHFR P00374 1/20 0.36
DHODH Q02127 1/20 0.36
ALKBH5 Q6P6C2 1/20 0.36
SCN2B O60939 1/20 0.35
SCN1B Q07699 1/20 0.35
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35
MAPT P10636 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3633770 0.89 NOTUM (0.41) NOTUMTP53NPC1GAARAB9A
SCHEMBL3634622 0.85 NOTUM (0.45) NOTUMTP53HSP90AA1PTGS1PTGS2
SCHEMBL3629591 0.84 ATM (0.46) TP53POLBGAAMAPTLMNA
SCHEMBL3633919 0.84 MEN1 (0.45) NOTUMGAA
SCHEMBL3633608 0.81 ABCB1 (0.53) NOTUMPTGS2LMNA
SCHEMBL3633758 0.81 NOTUM (0.44) NOTUMPTGS2SCN2BSCN1BSCN5A
SCHEMBL3631491 0.78 ABCB1 (0.49) NOTUMTP53POLBLMNAHTT
SCHEMBL3626683 0.78 NOTUM (0.42) NOTUMHSP90AA1GAARAB9AALKBH5
SCHEMBL3631115 0.76 CA12 (0.43) NOTUMTP53POLBNPC1RAB9A
SCHEMBL4283426 0.76 GRM1 (0.40) HTTTUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2010-02-10 EP disclosed
WO-2008131779-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2008-11-06 WO disclosed