SCHEMBL3633608

SCHEMBL3633608

Cc1c(C(=O)O)c2cc(=O)ccc-2cn1-c1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.53
NOTUM Q6P988 1/20 0.41
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GABRA2 P47869 1/20 0.38
GABRB2 P47870 1/20 0.38
HMGCR P04035 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CHRNA7 P36544 2/20 0.35
BCL2L1 Q07817 1/20 0.34
BAD Q92934 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3631491 0.90 ABCB1 (0.49) ABCB1NOTUMLMNAKDM4EL3MBTL1
SCHEMBL3633919 0.88 MEN1 (0.45) ABCB1NOTUMKDM4EMEN1KMT2A
SCHEMBL3631115 0.87 CA12 (0.43) ABCB1NOTUMLMNAKDM4EGABRA2
SCHEMBL3633758 0.86 NOTUM (0.44) ABCB1NOTUML3MBTL1MEN1KMT2A
SCHEMBL3631637 0.85 LMNA (0.43) LMNAKDM4EGABRA2GABRB2MEN1
SCHEMBL3633448 0.82 NOTUM (0.43) ABCB1NOTUMLMNAGABRA2GABRB2
SCHEMBL3632665 0.82 ABCB1 (0.50) ABCB1NOTUMLMNAKDM4EGABRA2
SCHEMBL3632144 0.81 ABCB1 (0.37) ABCB1NOTUMLMNAKDM4EGABRA2
SCHEMBL3626683 0.81 NOTUM (0.42) ABCB1NOTUMLMNAKDM4EL3MBTL1
SCHEMBL3631359 0.81 NOTUM (0.45) NOTUMLMNAPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2010-02-10 EP disclosed
WO-2008131779-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2008-11-06 WO disclosed