SCHEMBL3633758

SCHEMBL3633758

Cc1c(C(=O)O)c2cc(=O)ccc-2cn1-c1cccc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.44
ALDH1A1 P00352 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ABCB1 P08183 1/20 0.39
PTGS2 P35354 1/20 0.37
SCN2B O60939 3/20 0.35
SCN1B Q07699 3/20 0.35
SCN5A Q14524 3/20 0.35
SCN9A Q15858 3/20 0.35
SCN1A P35498 2/20 0.35
TSHR P16473 1/20 0.35
GRM1 Q13255 1/20 0.35
FAAH O00519 1/20 0.35
MGLL Q99685 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3626683 0.88 NOTUM (0.42) NOTUMALDH1A1L3MBTL1ABCB1GRM1
SCHEMBL3633919 0.87 MEN1 (0.45) NOTUMALDH1A1ABCB1MEN1KMT2A
SCHEMBL3633608 0.86 ABCB1 (0.53) NOTUML3MBTL1ABCB1PTGS2MEN1
SCHEMBL3632701 0.85 KDM4E (0.47) NOTUMALDH1A1TSHRMGLLMEN1
SCHEMBL3633358 0.83 NOTUM (0.44) NOTUMALDH1A1L3MBTL1ABCB1SCN2B
SCHEMBL3631491 0.81 ABCB1 (0.49) NOTUMALDH1A1L3MBTL1ABCB1MEN1
SCHEMBL4283426 0.81 GRM1 (0.40) ALDH1A1GRM1TUBB4ATUBBTUBA3C
SCHEMBL3631359 0.81 NOTUM (0.45) NOTUMPTGS2SCN2BSCN1BSCN5A
SCHEMBL3633448 0.80 NOTUM (0.43) NOTUMALDH1A1ABCB1
SCHEMBL3631115 0.79 CA12 (0.43) NOTUMALDH1A1ABCB1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2010-02-10 EP disclosed
WO-2008131779-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2008-11-06 WO disclosed