SCHEMBL363181

SCHEMBL363181

CC(=O)C(c1ccc(Br)cc1)(c1ccnc(C)c1)c1ccc(Cl)cc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CYP3A4 P08684 5/20 0.36
CYP3A5 P20815 5/20 0.36
KMO O15229 1/20 0.35
PROKR1 Q8TCW9 1/20 0.33
MAPK1 P28482 1/20 0.32
SORT1 Q99523 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KCNH2 Q12809 1/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
CCR9 P51686 1/20 0.31
KCNN4 O15554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362323 0.89 KCNN4 (0.41) HDAC3HDAC1HDAC2HDAC6KMO
SCHEMBL363084 0.89 SORT1 (0.34) PROKR1MAPK1SORT1ALDH1A1KCNH2
SCHEMBL364587 0.89 SORT1 (0.34) PROKR1MAPK1SORT1ALDH1A1KCNH2
SCHEMBL362712 0.89 SORT1 (0.34) PROKR1MAPK1SORT1ALDH1A1KCNH2
SCHEMBL364151 0.87 CYP3A4 (0.35) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL364096 0.87 CYP3A4 (0.35) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL364634 0.79 PROKR1 (0.35) PROKR1MAPK1SORT1KCNH2PSEN1
SCHEMBL364536 0.79 SORT1 (0.35) CYP3A4KMOSORT1ALDH1A1PSEN1
SCHEMBL363549 0.78 NPC1 (0.34) CYP3A4MAPK1SORT1ALDH1A1
SCHEMBL364193 0.78 NPC1 (0.34) CYP3A4MAPK1SORT1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed