SCHEMBL363183

SCHEMBL363183

Cc1cc(C(CC=O)(c2cccc(S(C)(=O)=O)c2)c2ccccc2C)ccn1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.36
NR1H2 P55055 9/20 0.35
NR1H3 Q13133 9/20 0.35
RXRA P19793 1/20 0.34
GRM5 P41594 1/20 0.34
JAK2 O60674 1/20 0.33
MAPK1 P28482 2/20 0.33
ALDH1A1 P00352 1/20 0.32
NR3C1 P04150 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.31
ROCK1 Q13464 1/20 0.31
LRRK2 Q5S007 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364731 0.88 KIF11 (0.34) KIF11NR1H2NR1H3RXRAGRM5
SCHEMBL15949082 0.80
SCHEMBL364417 0.80
SCHEMBL364334 0.78 NR1H2 (0.41) KIF11NR1H2NR1H3RXRA
SCHEMBL364292 0.76 NR1H2 (0.34) KIF11NR1H2NR1H3RXRAGRM5
SCHEMBL370168 0.75 CYP19A1 (0.33) KIF11
SCHEMBL363791 0.73 AHR (0.37) ALDH1A1
SCHEMBL363561 0.73 AHR (0.37) ALDH1A1
SCHEMBL362361 0.72 GPBAR1 (0.31) KIF11
SCHEMBL364428 0.71 IDH1 (0.31) RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed