SCHEMBL364334

SCHEMBL364334

Cc1cc(C(CC=O)(c2ccc(-c3ccc(S(C)(=O)=O)cc3)cc2)c2ccccc2C(F)(F)F)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 7/20 0.41
KIF11 P52732 1/20 0.40
NR1H3 Q13133 5/20 0.39
RORC P51449 1/20 0.39
SYK P43405 1/20 0.38
CYP2D6 P10635 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
FLT3 P36888 1/20 0.36
PTGS2 P35354 6/20 0.36
PTGS1 P23219 2/20 0.36
RXRA P19793 1/20 0.36
MAP4K4 O95819 1/20 0.35
PIK3CA P42336 1/20 0.35
KCNH2 Q12809 1/20 0.35
MINK1 Q8N4C8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365421 0.89 NR1H2 (0.39) NR1H2KIF11NR1H3RORCSYK
SCHEMBL362569 0.83 RORA (0.32)
SCHEMBL363183 0.78 KIF11 (0.36) NR1H2KIF11NR1H3RXRA
SCHEMBL363922 0.77 NR1H2 (0.41) NR1H2KIF11NR1H3RORCSYK
SCHEMBL15949082 0.73
SCHEMBL364417 0.73
SCHEMBL363663 0.71 CYP1A1 (0.33) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL364800 0.71 PDK2 (0.30)
SCHEMBL363668 0.70 RORC (0.40) RORCSYK
SCHEMBL370168 0.68 CYP19A1 (0.33) KIF11MAP4K4KCNH2MINK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed