SCHEMBL3632173

SCHEMBL3632173

N#CN=C(N)c1cc(F)ccc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.46
CES1 P23141 3/20 0.46
POLB P06746 1/20 0.43
CA3 P07451 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
KEAP1 Q14145 1/20 0.34
GRIN2D O15399 2/20 0.34
GRIN3B O60391 2/20 0.34
GRIN1 Q05586 2/20 0.34
GRIN2A Q12879 2/20 0.34
GRIN2B Q13224 2/20 0.34
GRIN2C Q14957 2/20 0.34
GRIN3A Q8TCU5 2/20 0.34
ALDH1A1 P00352 3/20 0.32
MDM2 Q00987 2/20 0.31
SLC9A1 P19634 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3632169 1.00 CES2 (0.46) CES2CES1POLBCA3CA6
SCHEMBL642417 0.77 CES2 (0.52) CES2CES1CA3CA6CA5A
SCHEMBL15489581 0.77 CES2 (0.52) CES2CES1CA3CA6CA5A
SCHEMBL642418 0.77 CES2 (0.52) CES2CES1CA3CA6CA5A
SCHEMBL12225512 0.77 CES2 (0.52) CES2CES1CA3CA6CA5A
Hydrochloric Acid SCHEMBL7963311 0.76 CES2 (0.50) CES2CES1CA3CA6CA5A
SCHEMBL4685491 0.71 ALDH1A1 (0.39) POLBCA3CA6CA5ACA9
SCHEMBL4685493 0.71 ALDH1A1 (0.39) POLBCA3CA6CA5ACA9
SCHEMBL3680333 0.69 CES2 (0.47) CES2CES1CA3CA6CA5A
SCHEMBL3680330 0.69 CES2 (0.47) CES2CES1CA3CA6CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2142522-A1 1, 3-THIAZOL-2 (3H) -YLIDENE COMPOUNDS AS CANNABINOID RECEPTOR LIGANDS Abbott Laboratories (US) 2010-01-13 EP claimed
WO-2008121558-A1 1, 3-THIAZOL-2 (3H) -YLIDENE COMPOUNDS AS CANNABINOID RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2008-10-09 WO claimed