SCHEMBL363679

SCHEMBL363679

Cc1cc(C(=O)O)ccc1-c1ccc(C(C/C(=N\O)c2c[nH]c(=O)c(C)c2)c2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.42
SRD5A2 P31213 2/20 0.41
ADRB1 P08588 3/20 0.39
ADRB3 P13945 3/20 0.39
SPR P35270 1/20 0.38
TNKS2 Q9H2K2 1/20 0.36
RARB P10826 1/20 0.35
MGAM O43451 1/20 0.34
GAA P10253 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
EIF4E P06730 1/20 0.34
CTSA P10619 1/20 0.33
MARS1 P56192 1/20 0.33
SLC1A3 P43003 1/20 0.33
SLC1A2 P43004 1/20 0.33
SLC1A1 P43005 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364066 1.00 GPBAR1 (0.42) GPBAR1SRD5A2ADRB1ADRB3SPR
SCHEMBL364024 1.00 GPBAR1 (0.42) GPBAR1SRD5A2ADRB1ADRB3SPR
SCHEMBL363638 0.92 GPBAR1 (0.41) GPBAR1SRD5A2ADRB1ADRB3SPR
SCHEMBL363248 0.92 GPBAR1 (0.41) GPBAR1SRD5A2ADRB1ADRB3SPR
SCHEMBL363277 0.92 GPBAR1 (0.41) GPBAR1SRD5A2ADRB1ADRB3SPR
SCHEMBL363178 0.87 GPBAR1 (0.51) GPBAR1SRD5A2ADRB1ADRB3SPR
SCHEMBL365274 0.86 GPBAR1 (0.46) GPBAR1SPRMGAMGAASI
SCHEMBL364353 0.84 GPBAR1 (0.47) GPBAR1TNKS2CTSAPRKAB2PRKAG1
SCHEMBL361680 0.84 GPBAR1 (0.47) GPBAR1SRD5A2ADRB1ADRB3SPR
SCHEMBL363787 0.84 GPBAR1 (0.38) GPBAR1ADRB1ADRB3SPRRARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed