SCHEMBL3634087

SCHEMBL3634087

CC(=O)C(Br)Cc1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.47
MME P08473 6/20 0.44
EPHX1 P07099 2/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP1A2 P05177 1/20 0.41
MAOB P27338 1/20 0.41
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31635698 0.84 ACACB (0.45) ACACBESR1ESR2MEN1KMT2A
SCHEMBL27986499 0.83 MME (0.45) ACACBMMEEPHX1MEN1NPC1
SCHEMBL4283538 0.82 SLC6A2 (0.47) ACACBESR1ESR2MEN1NPC1
SCHEMBL3713994 0.82 ALPI (0.53) NPC1RAB9ACYP1A2
SCHEMBL27807869 0.82 MME (0.51) MMEMEN1NPC1RAB9AKMT2A
SCHEMBL12459110 0.82 MME (0.53) ACACBMMEMEN1NPC1RAB9A
SCHEMBL1867578 0.82 ACACB (0.49) ACACBMMEEPHX1ESR1ESR2
SCHEMBL19369764 0.80 ACACB (0.47) ACACBMMEEPHX1ESR1ESR2
SCHEMBL14559931 0.80 SLC7A5 (0.48) ACACBMMEEPHX1ESR1ESR2
SCHEMBL14355742 0.80 SLC7A5 (0.48) ACACBMMEEPHX1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152271-A1 PIPERIDINE/PIPERAZINE DERIVATIVES Janssen Pharmaceutica, N.V. (BE) 2010-02-17 EP disclosed
WO-2008148840-A1 PIPERIDINE/PIPERAZINE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 2008-12-11 WO disclosed