SCHEMBL3634633

SCHEMBL3634633

COC(=O)CC(=O)Cc1cccc([N+](=O)[O-])c1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PDGFRB P09619 1/20 0.40
FGFR1 P11362 1/20 0.40
PDGFRA P16234 1/20 0.40
FLT1 P17948 1/20 0.40
FGFR3 P22607 1/20 0.40
KDR P35968 1/20 0.40
PTPN1 P18031 1/20 0.40
MAPT P10636 1/20 0.40
LMNA P02545 1/20 0.40
PLK1 P53350 1/20 0.40
PLK3 Q9H4B4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11872916 0.81 TDP1 (0.59) L3MBTL1TDP1TSHRSMN1; SMN2ALDH1A1
SCHEMBL5460845 0.80 TDP1 (0.57) L3MBTL1TDP1TSHRSMN1; SMN2ALDH1A1
SCHEMBL17336305 0.79 TDP1 (0.65) L3MBTL1TDP1TSHRSMN1; SMN2ALDH1A1
SCHEMBL3633747 0.79 CA12 (0.57) L3MBTL1MEN1KMT2ANPC1RAB9A
SCHEMBL3631412 0.79 ALDH1A1 (0.41) SMN1; SMN2ALDH1A1KMT2ALMNA
SCHEMBL20185133 0.77 L3MBTL1 (0.57) L3MBTL1TDP1TSHRSMN1; SMN2ALDH1A1
SCHEMBL4099366 0.76 TDP1 (0.50) L3MBTL1TDP1TSHRSMN1; SMN2ALDH1A1
SCHEMBL8477526 0.76 TDP1 (0.60) L3MBTL1TDP1TSHRALDH1A1PTPN1
SCHEMBL8477522 0.76 TDP1 (0.60) L3MBTL1TDP1TSHRALDH1A1PLK1
SCHEMBL6949395 0.76 PTPN1 (0.48) L3MBTL1TSHRSMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2010-02-10 EP disclosed
WO-2008131779-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2008-11-06 WO disclosed