SCHEMBL3635304

SCHEMBL3635304

CCCCC(=O)C=C(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.48
CES2 O00748 5/20 0.48
ALDH1A1 P00352 3/20 0.44
TP53 P04637 1/20 0.44
TRPA1 O75762 1/20 0.43
CA1 P00915 1/20 0.42
AKR1B1 P15121 1/20 0.39
POLB P06746 1/20 0.38
POLA1 P09884 1/20 0.38
HSP90AA1 P07900 1/20 0.38
IAPP P10997 1/20 0.38
PPARG P37231 3/20 0.37
PPARA Q07869 3/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 1/20 0.37
SLC22A6 Q4U2R8 1/20 0.37
SLC22A8 Q8TCC7 1/20 0.37
GPR84 Q9NQS5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL454224 0.93 TRPA1 (0.52) CES1CES2ALDH1A1TRPA1AKR1B1
SCHEMBL17867061 0.91 CES2 (0.52) CES1CES2ALDH1A1TRPA1POLB
Ammonia Solution, Strong SCHEMBL27538867 0.91 TRPA1 (0.50) CES1CES2ALDH1A1TRPA1AKR1B1
SCHEMBL4422427 0.91 CES2 (0.52) CES1CES2ALDH1A1TRPA1POLB
SCHEMBL11747932 0.91 CES2 (0.52) CES1CES2ALDH1A1TRPA1POLB
SCHEMBL11746072 0.91 CES2 (0.52) CES1CES2ALDH1A1TRPA1POLB
SCHEMBL3912771 0.91 CES2 (0.52) CES1CES2ALDH1A1TRPA1POLB
Oxalic Acid SCHEMBL1013866 0.87 AKR1B1 (0.48) CES1CES2ALDH1A1TRPA1AKR1B1
SCHEMBL4391467 0.84
SCHEMBL19599290 0.83 CES1 (0.46) CES1CES2ALDH1A1TP53TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5331086-A Deashing process for polyolefins using an alpha,beta-unsaturated ketone PHILLIPS PETROLEUM COMPANY (US) 1994-07-19 US claimed
EP-2930179-B1 RUTHENIUM COMPLEX AND METHOD FOR PRODUCING SAME, AND METHOD FOR PRODUCING RUTHENIUM-CONTAINING THIN FILM TOSOH CORP (JP) 2018-09-05 EP disclosed
US-20170210729-A1 ERK INHIBITORS AND USES THEREOF BRISTOL-MYERS SQUIBB COMPANY 2017-07-27 US disclosed
US-9694086-B2 HCV protease inhibitors and uses thereof CELGENE CAR LLC (BM) 2017-07-04 US disclosed
US-20160368930-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2016-12-22 US disclosed
US-20160326216-A1 HCV PROTEASE INHIBITORS AND USES THEREOF CELGENE CAR LLC (BM) 2016-11-10 US disclosed
US-20160243249-A1 HCV PROTEASE INHIBITORS AND USES THEREOF CELGENE CAR LLC (BM) 2016-08-25 US disclosed
US-9349601-B2 Ruthenium complex, method for producing same, and method for producing ruthenium-containing thin film TOSOH CORPORATION (JP) 2016-05-24 US disclosed
US-20160137610-A1 Compounds that Modulate EGFR Activity and Methods for Treating or Preventing Conditions Therewith Gatekeeper Pharmaceuticals, Inc. 2016-05-19 US disclosed
US-9296737-B2 Substituted 2,4-diaminopyrimidines as kinase inhibitors CELGENE AVILOMICS RESEARCH, INC. (US) 2016-03-29 US disclosed
WO-2008152086-A2 4,5-DIHYDRO-(1H)-PYRAZOLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR MODULATORS SOLVAY PHARMACEUTICALS B.V. (NL) 2008-12-18 WO disclosed
US-5331086-A Deashing process for polyolefins using an alpha,beta-unsaturated ketone PHILLIPS PETROLEUM COMPANY (US) 1994-07-19 US disclosed
EP-0073301-B1 PROCESS FOR THE PREPARATION OF ALPHA, BETA AND BETA, GAMMA UNSATURATED KETONES FIRMENICH SA (CH) 1984-11-21 EP disclosed
US-4453011-A BASIFICATION OF A DIALLYL CARBINOL FIRMENICH SA (CH) 1984-06-05 US disclosed
EP-0073301-A1 Process for the preparation of alpha, beta and beta, gamma unsaturated ketones FIRMENICH SA (CH) 1983-03-09 EP disclosed
US-4226892-A Flavoring with cycloaliphatic unsaturated ketones FIRMENICH SA (CH) 1980-10-07 US disclosed
US-4187863-A Cycloaliphatic unsaturated ketones as odor and taste modifying agents in tobacco products FIRMENICH SA (CH) 1980-02-12 US disclosed
US-4002684-A FROM AN ALPHA,BETA-UNSATURATED KETONE AND A VINYLMAGNESIUM HALIDE, COPPER COMPOUND CATALYST BASF AKTIENGESELLSCHAFT (DT) 1977-01-11 US disclosed
US-3975310-A PERFUME FIRMENICH S.A. (CH) 1976-08-17 US disclosed
US-3931326-A FLAVOR, TASTE, ODOR, PERFUMES FIRMENICH SA (CH) 1976-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160137610-A1 Compounds that Modulate EGFR Activity and Methods for Treating or Preventing Conditions Therewith EGFR, ERBB2, BRCA1 CES1 567/4885CES2 1157/4885ALDH1A1 2351/4885
US-20160243249-A1 HCV PROTEASE INHIBITORS AND USES THEREOF PEPD, CTRL, CTSC CES1 76/4885CES2 145/4885ALDH1A1 1344/4885
US-20160326216-A1 HCV PROTEASE INHIBITORS AND USES THEREOF PEPD, CTRL, CTSC CES1 76/4885CES2 145/4885ALDH1A1 1344/4885
US-20160368930-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER KRAS, HRAS, NRAS CES1 3108/4885CES2 4000/4885ALDH1A1 2792/4885
US-20170210729-A1 ERK INHIBITORS AND USES THEREOF MAP3K20, MAP3K1, MAPK3 CES1 3085/4885CES2 3619/4885ALDH1A1 2838/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.