SCHEMBL363663

SCHEMBL363663

Cc1cc(C(CC=O)(c2ccc(C(F)(F)F)cc2)c2ccc(F)cc2F)ccn1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
CYP3A4 P08684 2/20 0.32
SORT1 Q99523 1/20 0.32
RXRA P19793 1/20 0.31
MAPK1 P28482 3/20 0.31
PSEN1 P49768 4/20 0.31
PSEN2 P49810 4/20 0.31
APH1B Q8WW43 4/20 0.31
NCSTN Q92542 4/20 0.31
APH1A Q96BI3 4/20 0.31
PSENEN Q9NZ42 4/20 0.31
CYP2D6 P10635 2/20 0.31
CYP3A5 P20815 1/20 0.31
PDE2A O00408 2/20 0.31
GRM2 Q14416 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362479 0.90 HDAC3 (0.30)
SCHEMBL363954 0.81 HDAC6 (0.32)
SCHEMBL364445 0.80 CYP3A4 (0.35) CYP3A4MAPK1CYP3A5
SCHEMBL364596 0.77
SCHEMBL362569 0.76 RORA (0.32) SORT1GRM2
SCHEMBL364740 0.71 KCNN4 (0.36) CYP1A1CYP1B1CYP3A4SORT1PSEN1
SCHEMBL364334 0.71 NR1H2 (0.41) RXRAPSEN1PSEN2APH1BNCSTN
SCHEMBL15949082 0.70
SCHEMBL364417 0.70
SCHEMBL363251 0.70 KCNH2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed