SCHEMBL363734

SCHEMBL363734

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)N[C@H](CO)C(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.45
BRD4 O60885 1/20 0.39
PAK4 O96013 1/20 0.35
CTSA P10619 6/20 0.34
TAS1R3 Q7RTX0 2/20 0.33
TAS1R1 Q7RTX1 2/20 0.33
GABRA5 P31644 1/20 0.33
SLC6A9 P48067 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ROCK2 O75116 3/20 0.32
ROCK1 Q13464 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363430 1.00 GPBAR1 (0.45) GPBAR1BRD4PAK4CTSATAS1R3
SCHEMBL361767 0.91 GPBAR1 (0.47) GPBAR1BRD4CTSATAS1R3TAS1R1
SCHEMBL362542 0.91 GPBAR1 (0.47) GPBAR1BRD4CTSATAS1R3TAS1R1
SCHEMBL363956 0.90 BRD4 (0.41) GPBAR1BRD4PAK4CTSATAS1R3
SCHEMBL370940 0.90 BRD4 (0.41) GPBAR1BRD4PAK4CTSATAS1R3
SCHEMBL364032 0.85 GPBAR1 (0.47) GPBAR1BRD4SLC6A9KDM4EMAPT
SCHEMBL362902 0.85 GPBAR1 (0.45) GPBAR1BRD4GABRA5SLC6A9KDM4E
SCHEMBL363678 0.85 GPBAR1 (0.61) GPBAR1BRD4CTSA
SCHEMBL364239 0.84 GPBAR1 (0.47) GPBAR1BRD4SLC6A9KDM4EMAPT
SCHEMBL363542 0.84 GPBAR1 (0.47) GPBAR1BRD4SLC6A9KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed