SCHEMBL364032

SCHEMBL364032

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)NCCO)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.47
BRD4 O60885 1/20 0.40
EPHX2 P34913 4/20 0.39
SLC6A9 P48067 1/20 0.36
LMNA P02545 3/20 0.34
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
SPHK2 Q9NRA0 1/20 0.34
SPHK1 Q9NYA1 1/20 0.34
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 2/20 0.34
MAPT P10636 2/20 0.34
MAPK1 P28482 2/20 0.34
KMT2A Q03164 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
MMP13 P45452 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364071 0.92 GPBAR1 (0.47) GPBAR1BRD4EPHX2
SCHEMBL363585 0.91 GPBAR1 (0.45) GPBAR1BRD4EPHX2MAPK1NPC1
SCHEMBL362350 0.90 GPBAR1 (0.48) GPBAR1BRD4EPHX2SLC6A9MAPT
SCHEMBL363032 0.90 GPBAR1 (0.45) GPBAR1BRD4EPHX2SLC6A9LMNA
SCHEMBL362795 0.89 GPBAR1 (0.36) GPBAR1BRD4EPHX2POLBALDH1A1
SCHEMBL362902 0.89 GPBAR1 (0.45) GPBAR1BRD4EPHX2SLC6A9LMNA
SCHEMBL363542 0.89 GPBAR1 (0.47) GPBAR1BRD4EPHX2SLC6A9LMNA
SCHEMBL364239 0.89 GPBAR1 (0.47) GPBAR1BRD4EPHX2SLC6A9LMNA
SCHEMBL363667 0.87 GPBAR1 (0.42) GPBAR1BRD4EPHX2ALDH1A1MAPT
SCHEMBL363678 0.87 GPBAR1 (0.61) GPBAR1BRD4L3MBTL1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed