SCHEMBL363678

SCHEMBL363678

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.61
BRD4 O60885 1/20 0.41
MGAM O43451 5/20 0.36
GAA P10253 5/20 0.36
SI P14410 5/20 0.36
MGAM2 Q2M2H8 5/20 0.36
CTSA P10619 2/20 0.33
HPGD P15428 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
TTR P02766 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362545 0.97 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL363349 0.97 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL364601 0.97 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL363650 0.90 GPBAR1 (0.58) GPBAR1BRD4MGAMGAASI
SCHEMBL364092 0.89 GPBAR1 (0.48) GPBAR1BRD4MGAMGAASI
SCHEMBL363444 0.88 GPBAR1 (0.55) GPBAR1BRD4MGAMGAASI
SCHEMBL362527 0.88 GPBAR1 (0.55) GPBAR1BRD4MGAMGAASI
SCHEMBL362350 0.88 GPBAR1 (0.48) GPBAR1BRD4CTSACYP3A4
SCHEMBL363934 0.87 GPBAR1 (0.47) GPBAR1BRD4MGAMGAASI
SCHEMBL365274 0.87 GPBAR1 (0.46) GPBAR1BRD4MGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed