SCHEMBL3637604

SCHEMBL3637604

O=c1[nH]c2ccccc2n1C1CCN(C2CCCN(Cc3ccccc3)C2)CC1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 8/20 0.73
OPRK1 P41145 1/20 0.73
OPRL1 P41146 1/20 0.73
CHRM1 P11229 5/20 0.66
CHRM2 P08172 3/20 0.66
CHRM4 P08173 3/20 0.66
CHRM3 P20309 2/20 0.66
ALDH1A1 P00352 1/20 0.61
TSHR P16473 1/20 0.61
MAPK1 P28482 1/20 0.61
DRD2 P14416 2/20 0.60
CHRM5 P08912 1/20 0.58
ADRA1D P25100 1/20 0.58
HTR2C P28335 1/20 0.58
ADRA1A P35348 1/20 0.58
ADRA1B P35368 1/20 0.58
DRD4 P21917 1/20 0.57
AKT1 P31749 1/20 0.56
AKT2 P31751 1/20 0.56
AKT3 Q9Y243 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8863557 0.88 OPRM1 (0.91) OPRM1OPRK1OPRL1CHRM1CHRM2
SCHEMBL11223608 0.88 OPRM1 (0.86) OPRM1OPRK1OPRL1CHRM1DRD4
SCHEMBL3665096 0.85 OPRM1 (1.00) OPRM1OPRK1OPRL1CHRM1DRD2
Oxalic Acid SCHEMBL5778025 0.83 OPRM1 (0.91) OPRM1OPRK1OPRL1ALDH1A1DRD2
SCHEMBL3630723 0.82 OPRM1 (0.66) OPRM1OPRK1OPRL1CHRM1CHRM2
SCHEMBL3895786 0.81 CHRM1 (0.92) OPRM1OPRK1OPRL1CHRM1CHRM2
SCHEMBL6487094 0.81 OPRM1 (0.61) OPRM1OPRK1OPRL1CHRM1CHRM2
SCHEMBL4919819 0.80 CHRM1 (1.00) OPRM1OPRK1OPRL1CHRM1CHRM2
SCHEMBL4572894 0.80 CHRM1 (1.00) OPRM1OPRK1OPRL1CHRM1CHRM2
SCHEMBL27056694 0.80 CHRM1 (1.00) OPRM1OPRK1OPRL1CHRM1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155676-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS Commissariat à l'Energie Atomique (FR) 2010-02-24 EP disclosed
WO-2008146172-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-12-04 WO disclosed