SCHEMBL3639596

SCHEMBL3639596

COC(=O)[C@@H]1C[C@@H](O)CN1Cc1cccc(Cl)c1.ClCc1cccc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MC3R P41968 1/20 0.42
MC1R Q01726 1/20 0.42
CYP3A4 P08684 2/20 0.42
VHL P40337 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CXCR6 O00574 1/20 0.39
CD274 Q9NZQ7 2/20 0.39
PDCD1 Q15116 1/20 0.39
OPRK1 P41145 1/20 0.39
MAPT P10636 1/20 0.39
MMP1 P03956 1/20 0.38
ADAM17 P78536 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2820776 0.95 MAOA (0.46) MAOAMAOBKDM4EMC3RMC1R
SCHEMBL2818883 0.83 CYP3A4 (0.50) MAOAMAOBKDM4ECYP3A4KMT2A
SCHEMBL4249938 0.83 CYP3A4 (0.50) MAOAMAOBKDM4ECYP3A4KMT2A
SCHEMBL1440329 0.83 CYP3A4 (0.50) MAOAMAOBKDM4ECYP3A4KMT2A
SCHEMBL15325590 0.83 CYP3A4 (0.50) MAOAMAOBKDM4ECYP3A4KMT2A
SCHEMBL24938939 0.83 CYP3A4 (0.50) MAOAMAOBKDM4ECYP3A4KMT2A
SCHEMBL5368566 0.83 CYP3A4 (0.50) MAOAMAOBKDM4ECYP3A4KMT2A
SCHEMBL19408855 0.83 CYP3A4 (0.50) MAOAMAOBKDM4ECYP3A4KMT2A
Hydrochloric Acid SCHEMBL6951431 0.82 CYP3A4 (0.49) MAOAMAOBKDM4ECYP3A4KMT2A
SCHEMBL2817870 0.80 ALDH1A1 (0.47) MAOAMAOBKDM4EMC3RMC1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155672-A1 PROLINAMIDE DERIVATIVES AS NK3 ANTAGONISTS F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008148689-A1 PROLINAMIDE DERIVATIVES AS NK3 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-12-11 WO disclosed