SCHEMBL3639809

SCHEMBL3639809

CCOC(=O)c1onc2cc(-c3ccc(O)cc3)ccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.46
ESR2 Q92731 2/20 0.46
CA12 O43570 4/20 0.44
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA7 P43166 4/20 0.44
CA9 Q16790 4/20 0.44
CA14 Q9ULX7 4/20 0.44
ROCK2 O75116 1/20 0.41
CDK1 P06493 1/20 0.41
PRKACA P17612 1/20 0.41
CDK2 P24941 1/20 0.41
CSNK1D P48730 1/20 0.41
GSK3A P49840 1/20 0.41
CDK5 Q00535 1/20 0.41
PRKCD Q05655 1/20 0.41
ROCK1 Q13464 1/20 0.41
CDC42BPA Q5VT25 1/20 0.41
MARK2 Q7KZI7 1/20 0.41
AKR1B1 P15121 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3635258 0.80 ALDH1A1 (0.49) ALDH1A1HTTTSHRSMN1; SMN2TARBP2
SCHEMBL6819286 0.80 KDM4E (0.48) ALDH1A1HPGDTSHRKDM4ESMN1; SMN2
SCHEMBL2815397 0.80 ESR1 (0.44) ESR1ESR2CA12CA1CA2
SCHEMBL6819051 0.77 ALDH1A1 (0.43) ALDH1A1HPGDTSHRKDM4ESMN1; SMN2
SCHEMBL6818394 0.76 KDM4E (0.51) ALDH1A1TSHRKDM4ESMN1; SMN2MEN1
SCHEMBL25170921 0.76 MAPT (0.39) ESR1ESR2CA12CA1CA2
SCHEMBL25171020 0.74 KDM4E (0.49) ALDH1A1HPGDKDM4ESMN1; SMN2MEN1
SCHEMBL17437927 0.74 CA12 (0.44) ESR2CA12CA1CA2CA7
SCHEMBL5985145 0.72 ALDH1A1 (0.55) ALDH1A1TSHRSMN1; SMN2MEN1KMT2A
SCHEMBL11972313 0.70 CA12 (0.53) ESR1ESR2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170072-A1 FARNESOID X RECEPTOR AGONISTS GlaxoSmithKline LLC (US) 2010-04-07 EP disclosed
WO-2008157270-A1 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed