SCHEMBL2815397

SCHEMBL2815397

CCOC(=O)c1noc2cc(-c3ccc(O)cc3)ccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.44
ESR2 Q92731 4/20 0.44
CA12 O43570 3/20 0.44
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA7 P43166 3/20 0.44
CA9 Q16790 3/20 0.44
CA14 Q9ULX7 3/20 0.44
AKR1B1 P15121 1/20 0.44
HTT P42858 1/20 0.43
ALOX5 P09917 2/20 0.42
MLYCD O95822 1/20 0.42
TARBP2 Q15633 2/20 0.41
ROCK2 O75116 1/20 0.41
CDK1 P06493 1/20 0.41
PRKACA P17612 1/20 0.41
CDK2 P24941 1/20 0.41
CSNK1D P48730 1/20 0.41
GSK3A P49840 1/20 0.41
CDK5 Q00535 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL492496 0.89 AKR1B1 (0.54) ESR1ESR2CA12CA1CA2
SCHEMBL2083597 0.87 ESR1 (0.51) ESR1ESR2CA12CA1CA2
SCHEMBL6821684 0.81 TDP1 (0.45) HTTALOX5MLYCDTARBP2KMT2A
SCHEMBL8226588 0.80 HTT (0.50) HTTMLYCDALDH1A1
SCHEMBL492231 0.80 TBK1 (0.48) HTTALOX5TARBP2ALDH1A1
SCHEMBL492601 0.80 LMNA (0.46) AKR1B1HTTMLYCDMEN1KMT2A
SCHEMBL6833807 0.80 ALDH1A1 (0.50) TARBP2KMT2AGAAALDH1A1HPGD
SCHEMBL14492918 0.80 KDM4E (0.42) AKR1B1HTTMLYCDTARBP2KMT2A
SCHEMBL3639809 0.80 ESR1 (0.46) ESR1ESR2CA12CA1CA2
SCHEMBL2816030 0.79 DUSP3 (0.53) ESR1ESR2HSP90AA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100249179-A1 Farnesoid X Receptor Agonists SMITHKLINE BEECHAM CORPORATION (US) 2010-09-30 US disclosed
US-20100249179-A1 Farnesoid X Receptor Agonists SMITHKLINE BEECHAM CORPORATION (US) 2010-09-30 US disclosed
US-20100249179-A1 Farnesoid X Receptor Agonists SMITHKLINE BEECHAM CORPORATION (US) 2010-09-30 US disclosed
WO-2008157270-A1 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100249179-A1 Farnesoid X Receptor Agonists NR1H4, NR1H3, NR1H2 ESR1 451/4885ESR2 251/4885CA12 4597/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.