SCHEMBL3645646

SCHEMBL3645646

NC(c1cccc(Oc2ccccc2)c1)[C@@H]1CCCN1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.50
SLC6A2 P23975 4/20 0.50
SLC6A4 P31645 4/20 0.50
PTGS1 P23219 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
DHFR P00374 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3647068 1.00 SLC6A3 (0.50) SLC6A3SLC6A2SLC6A4PTGS1OPRM1
SCHEMBL28809365 0.82 SLC6A3 (0.50) SLC6A3SLC6A2SLC6A4DHFR
SCHEMBL4158218 0.82 SLC6A3 (0.50) SLC6A3SLC6A2SLC6A4DHFR
SCHEMBL4156194 0.82 SLC6A3 (0.50) SLC6A3SLC6A2SLC6A4DHFR
SCHEMBL17169355 0.78 SLC6A3 (0.56) SLC6A3SLC6A2SLC6A4DHFR
SCHEMBL4307731 0.73 LTA4H (0.46) SLC6A3SLC6A2SLC6A4
SCHEMBL27996273 0.72 SLC6A3 (0.52) SLC6A3SLC6A2SLC6A4DHFR
Proline SCHEMBL5760690 0.72 HTR2C (0.42) PTGS1
Hydrochloric Acid SCHEMBL4313825 0.71 SLC6A3 (0.51) SLC6A3SLC6A2SLC6A4DHFR
Hydrochloric Acid SCHEMBL4313832 0.71 SLC6A3 (0.51) SLC6A3SLC6A2SLC6A4DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183216-A1 2-AZETIDINEMETHANEAMINES AND 2-PYRROLIDINEMETHANEAMINES AS TAAR-LIGANDS F. Hoffmann-Roche AG (CH) 2010-05-12 EP disclosed
WO-2009016048-A1 2-AZETIDINEMETHANEAMINES AND 2-PYRROLIDINEMETHANEAMINES AS TAAR-LIGANDS F. HOFFMANN-LA ROCHE AG (CH) 2009-02-05 WO disclosed