SCHEMBL3646366

SCHEMBL3646366

Fc1cccc(-c2[c]c(C(F)(F)F)on2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.39
CYP11B2 P19099 2/20 0.38
NOTUM Q6P988 2/20 0.37
NT5E P21589 2/20 0.37
GRM5 P41594 2/20 0.37
HTR7 P34969 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP11B1 P15538 1/20 0.36
MGAM O43451 1/20 0.35
GAA P10253 1/20 0.35
SI P14410 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
HDAC4 P56524 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
ESR2 Q92731 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3645802 0.82 S1PR1 (0.40) NOTUMESR2
SCHEMBL27936742 0.81 TP53 (0.41) TP53CYP11B2NOTUMGRM5HTR7
SCHEMBL16104094 0.70 HDAC6 (0.61) TP53HDAC1HDAC8HDAC6HDAC4
SCHEMBL3150963 0.69 MEN1 (0.38) TP53NOTUMESR2
SCHEMBL2320359 0.68 MEN1 (0.47) TP53CYP11B2NOTUMNT5EGRM5
SCHEMBL11593511 0.65 PTGS1 (0.51) TP53NOTUMHTR7MGAMGAA
SCHEMBL198702 0.64 TAAR1 (0.68) CYP11B2NOTUMCYP17A1CYP3A4CYP11B1
SCHEMBL16877278 0.64 KDM4E (0.39) CYP11B2CYP17A1CYP3A4CYP11B1MGAM
SCHEMBL24799555 0.64 RPS6KB1 (0.52) TP53NOTUMCYP3A4MGAMGAA
SCHEMBL15219993 0.64 NPC1 (0.47) TP53NOTUMGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170873-A1 ISOXAZOLE-IMIDAZOLE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-04-07 EP disclosed
WO-2009000662-A1 ISOXAZOLE-IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-12-31 WO disclosed