SCHEMBL364699

SCHEMBL364699

Cc1cc(C(CC=O)(c2ccccc2)c2ccccc2)cc(C)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.35
EDNRB P24530 6/20 0.34
EDNRA P25101 6/20 0.34
RECQL P46063 1/20 0.34
NR1I2 O75469 1/20 0.34
KCNE1 P15382 1/20 0.34
KCNQ1 P51787 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
KIF11 P52732 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.33
CYP1A2 P05177 1/20 0.33
DHODH Q02127 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363298 0.90 EGFR (0.32) GAAMAPTTSHREDNRBEDNRA
SCHEMBL440368 0.82 KIF11 (0.41) TSHRKMT2AKIF11CYP2C19CYP1A2
SCHEMBL362227 0.80 EDNRB (0.33) GAAMAPTEDNRBEDNRANR1I2
SCHEMBL363076 0.71 EDNRB (0.30) EDNRBEDNRA
SCHEMBL10144369 0.70 CYP1A2 (0.42) GAAMAPTTSHREDNRBEDNRA
SCHEMBL363777 0.68 KMT2A (0.39) MAPTTSHRPOLBKMT2AKIF11
SCHEMBL369625 0.67 EDNRB (0.34) GAAMAPTTSHREDNRBEDNRA
SCHEMBL9340359 0.66 CYP2C19 (0.42) MAPTTSHRKMT2ACYP3A4CYP2D6
SCHEMBL6991557 0.66 CYP2C9 (0.44) TSHRKMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL1125158 0.66 TAAR1 (0.52) MAPTTSHRKMT2ACYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed