SCHEMBL3649821

SCHEMBL3649821

CN(Cc1cc(-c2cccnc2F)c(Br)s1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.38
SOS1 Q07889 1/20 0.38
PDK2 Q15119 1/20 0.37
HTR2C P28335 8/20 0.35
SLC6A4 P31645 8/20 0.35
GLS O94925 3/20 0.35
CACNA1G O43497 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNA1C Q13936 1/20 0.34
HTR2A P28223 1/20 0.34
TACR1 P25103 2/20 0.33
P2RY1 P47900 1/20 0.31
KCNH2 Q12809 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654912 0.85 CLK1 (0.32) SOS1PDK2
SCHEMBL4131558 0.85 AR (0.36) TACR1AR
SCHEMBL3652258 0.83 SSTR4 (0.38) SSTR4SOS1PDK2HTR2CSLC6A4
SCHEMBL3652077 0.83 SOS1 (0.36) SSTR4SOS1PDK2HTR2CSLC6A4
SCHEMBL3652574 0.82 HTR2C (0.35) SSTR4SOS1PDK2HTR2CSLC6A4
SCHEMBL3654372 0.82 HTR2C (0.34) SSTR4SOS1PDK2HTR2CSLC6A4
SCHEMBL3654948 0.81 F2 (0.35) SOS1PDK2HTR2CSLC6A4GLS
SCHEMBL3649951 0.81 PDK2 (0.35) SOS1PDK2HTR2CSLC6A4GLS
SCHEMBL3654413 0.81 HTR2C (0.33) SSTR4SOS1PDK2HTR2CSLC6A4
SCHEMBL3645627 0.81 CTSD (0.38) SSTR4PDK2HTR2CSLC6A4GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed