SCHEMBL3652258

SCHEMBL3652258

CN(Cc1nc(-c2cccnc2F)c(Br)s1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.38
SOS1 Q07889 1/20 0.38
PDK2 Q15119 1/20 0.37
CACNA1G O43497 1/20 0.36
CACNA1B Q00975 1/20 0.36
CACNA1C Q13936 1/20 0.36
GLS O94925 3/20 0.35
GBA1 P04062 1/20 0.34
HTR2C P28335 5/20 0.33
SLC6A4 P31645 5/20 0.33
TACR1 P25103 2/20 0.33
ROCK2 O75116 1/20 0.33
HTR2A P28223 1/20 0.33
PAX8 Q06710 1/20 0.32
DHODH Q02127 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3652850 0.87 SOS1 (0.39) SSTR4SOS1PDK2CACNA1GCACNA1B
SCHEMBL3649570 0.86 HTR6 (0.34) SOS1PDK2CACNA1GCACNA1BCACNA1C
SCHEMBL4118030 0.86 DHODH (0.36) TACR1ROCK2DHODHHDAC1HDAC6
SCHEMBL3655557 0.84 HTR2C (0.35) SSTR4SOS1PDK2CACNA1GCACNA1B
SCHEMBL3649821 0.83 SSTR4 (0.38) SSTR4SOS1PDK2CACNA1GCACNA1B
SCHEMBL3653351 0.83 GBA1 (0.35) SOS1PDK2CACNA1GCACNA1BCACNA1C
SCHEMBL3648527 0.81 ABCC9 (0.35) SOS1PDK2CACNA1GCACNA1BCACNA1C
SCHEMBL3780114 0.80 DHODH (0.31) TACR1ROCK2DHODH
SCHEMBL3654453 0.80 L3MBTL1 (0.36) SSTR4PDK2CACNA1GCACNA1BCACNA1C
SCHEMBL3652596 0.80 CACNA1G (0.34) SSTR4SOS1PDK2CACNA1GCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed