SCHEMBL3649825

SCHEMBL3649825

CC(C)(C)C(Cc1cc(-c2cccnc2F)c(Br)s1)NC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.34
DHODH Q02127 4/20 0.32
LIPG Q9Y5X9 3/20 0.31
LIPC P11150 1/20 0.31
CHRM4 P08173 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
NAPRT Q6XQN6 1/20 0.31
WNT1 P04628 1/20 0.31
GRIN3B O60391 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2C Q14957 1/20 0.30
ABL1 P00519 1/20 0.30
GSK3B P49841 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654915 0.85 GSK3B (0.33) DHODHGSK3BKMT2A
SCHEMBL4023651 0.83 DYRK1A (0.33) DYRK1ALIPG
SCHEMBL3652261 0.83 DHODH (0.35) DYRK1ADHODHLIPGLIPCCHRM4
SCHEMBL3652576 0.82 DYRK1A (0.34) DYRK1ADHODHCYP2D6KMT2A
SCHEMBL3804665 0.82 DYRK1A (0.34) DYRK1ALIPGLIPC
SCHEMBL3654414 0.81 DYRK1A (0.34) DYRK1A
SCHEMBL3649952 0.81 ABCC9 (0.36) LIPGLIPCKMT2A
SCHEMBL3654949 0.81 AGTR2 (0.33) LIPGLIPC
SCHEMBL3650566 0.81 DYRK1A (0.33) DYRK1A
SCHEMBL3645628 0.80 DYRK1A (0.40) DYRK1ADHODHLIPGLIPCCHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed