SCHEMBL3650759

SCHEMBL3650759

O=[N+]([O-])c1cc(S(=O)(=O)N2CCN(c3nc(Cc4cc(F)cc(Cl)c4)cs3)CC2)ccc1Cl.O=[N+]([O-])c1cc(S(=O)(=O)N2CCN(c3nc(Cc4ccc(F)c(Cl)c4)cs3)CC2)ccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 3/20 0.43
CYP17A1 P05093 1/20 0.42
CYP21A2 P08686 1/20 0.42
CYP11B1 P15538 1/20 0.42
NPBWR1 P48145 1/20 0.42
MCHR1 Q99705 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.40
ALDH1A1 P00352 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 5/20 0.39
LMNA P02545 2/20 0.39
MITF O75030 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
USP2 O75604 1/20 0.36
RECQL P46063 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GBA1 P04062 1/20 0.35
PIK3CD O00329 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3016494 0.95 VCAM1 (0.47) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1
SCHEMBL3019772 0.94 VCAM1 (0.48) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1
SCHEMBL3649645 0.93 VCAM1 (0.46) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1
SCHEMBL2998933 0.91 VCAM1 (0.49) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1
SCHEMBL3015121 0.90 VCAM1 (0.48) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1
SCHEMBL3019766 0.90 VCAM1 (0.51) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1
SCHEMBL3013323 0.89 VCAM1 (0.48) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1
SCHEMBL3008545 0.89 ALDH1A1 (0.48) SMN1; SMN2ALDH1A1L3MBTL1MAPTLMNA
SCHEMBL3007276 0.88 VCAM1 (0.51) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1
SCHEMBL3012868 0.86 VCAM1 (0.51) VCAM1CYP17A1CYP21A2CYP11B1NPBWR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188272-A2 PHENYL- AND BENZYLTHIAZOLYLPIPERAZINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES NV Remynd (BE) 2010-05-26 EP disclosed
WO-2009019295-A2 PHENYL- AND BENZYLTHIAZOLYLPIPERAZINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES NV REMYND (BE) 2009-02-12 WO disclosed