SCHEMBL3653137

SCHEMBL3653137

O=C(NC1CCCCC1)C(C1CCCCC1)C1(CCCOc2ccccc2)Nc2cc(F)c(Cl)cc2N1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P4HB P07237 1/20 0.40
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
RAB9A P51151 4/20 0.37
NPC1 O15118 3/20 0.37
CYP3A4 P08684 1/20 0.37
KCNH2 Q12809 1/20 0.37
NR1H4 Q96RI1 1/20 0.37
ALDH1A1 P00352 4/20 0.36
LMNA P02545 3/20 0.36
KDM4E B2RXH2 1/20 0.36
ALOX12 P18054 1/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
PKM P14618 1/20 0.35
EPHX2 P34913 1/20 0.35
METAP2 P50579 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3651703 0.89 NR1H4 (0.42) P4HBMEN1KMT2ARAB9ANPC1
SCHEMBL3649388 0.88 MEN1 (0.40) P4HBMEN1KMT2ARAB9ANPC1
SCHEMBL2907586 0.84 EPHX1 (0.41) MEN1KMT2ARAB9ANPC1CYP3A4
SCHEMBL3650434 0.84 KMT2A (0.41) MEN1KMT2ARAB9ANPC1ALDH1A1
SCHEMBL3649241 0.83 NR1H4 (0.45) KMT2ARAB9ANPC1CYP3A4KCNH2
SCHEMBL3651507 0.82 RAB9A (0.44) MEN1KMT2ARAB9ANPC1ALDH1A1
SCHEMBL3652035 0.81 EPHX2 (0.47) MEN1KMT2ARAB9ANPC1ALDH1A1
SCHEMBL3652322 0.80 CYP3A4 (0.37) MEN1KMT2ARAB9ANPC1CYP3A4
SCHEMBL3654059 0.79 EPHX1 (0.44) MEN1KMT2ARAB9ANPC1ALDH1A1
SCHEMBL3653797 0.79 RAB9A (0.45) MEN1KMT2ARAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188263-A1 BENZIMIDAZOLE DERIVATIVES USED AS FXR AGONISTS F. Hoffmann-Roche AG (CH) 2010-05-26 EP disclosed
WO-2009027264-A1 BENZIMIDAZOLE DERIVATIVES USED AS FXR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-03-05 WO disclosed