SCHEMBL365348

SCHEMBL365348

CS(=O)(=O)NC(=O)c1ccc(OCc2ccc(Cl)c(F)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 10/20 0.56
SCN5A Q14524 1/20 0.54
MAOB P27338 2/20 0.52
MAOA P21397 1/20 0.52
MRGPRX4 Q96LA9 1/20 0.51
KCNH2 Q12809 1/20 0.46
BCL2L1 Q07817 4/20 0.45
MCL1 Q07820 4/20 0.45
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364950 0.89 MAOB (0.66) SCN9ASCN5AMAOBMAOAMRGPRX4
SCHEMBL10203178 0.89 SCN9A (0.66) SCN9ASCN5AMAOBMAOAMRGPRX4
SCHEMBL16240196 0.84 SCN9A (0.77) SCN9ASCN5AMRGPRX4BCL2L1MCL1
SCHEMBL364615 0.83 MAOA (0.51) SCN9ASCN5AMAOBMAOAMRGPRX4
SCHEMBL365210 0.83 MAOA (0.63) SCN9ASCN5AMAOBMAOABCL2L1
SCHEMBL366081 0.83 MAOA (0.63) SCN9ASCN5AMAOBMAOABCL2L1
SCHEMBL366812 0.83 MAOB (0.63) SCN9AMAOBBCL2L1MCL1ALDH1A1
SCHEMBL367348 0.82 BCL2L1 (0.57) SCN9ASCN5AMAOBMAOAMRGPRX4
SCHEMBL14890621 0.82 GSK3B (0.55) SCN9ASCN5AMAOBBCL2L1MCL1
SCHEMBL679943 0.82 SCN9A (0.57) SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
EP-2593428-A2 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS Pfizer Limited (GB) 2013-05-22 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A SCN9A 16/4885SCN5A 5/4885MAOB 3660/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.