SCHEMBL3655949

SCHEMBL3655949

Cc1ccc(-c2c(C#N)c(NCCCOCCN(C)C)nc3sc(OC(N)=O)c(N)c23)o1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
MAPT P10636 3/20 0.34
HPGD P15428 2/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
HSP90AB1 P08238 1/20 0.31
PKM P14618 1/20 0.31
LIMK1 P53667 1/20 0.30
MAPK8 P45983 1/20 0.30
MAPK9 P45984 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3649451 0.93 ALDH1A1 (0.37) ALDH1A1MAPTHPGDMEN1GAA
SCHEMBL3101686 0.90 MAPT (0.46) ALDH1A1MAPTHPGDMEN1GAA
SCHEMBL3656735 0.89 MAPT (0.39) ALDH1A1MAPTHPGDMEN1GAA
SCHEMBL3657321 0.87 EEF2K (0.36) ALDH1A1KDM4EHSD17B10MAPK8MAPK9
SCHEMBL3649435 0.87 ALDH1A1 (0.38) ALDH1A1MAPTHPGDMEN1GAA
SCHEMBL3655988 0.84 ALDH1A1 (0.36) ALDH1A1MAPTHPGDMEN1GAA
SCHEMBL3657488 0.84 EEF2K (0.35) ALDH1A1KDM4EHSD17B10TLR7PKM
SCHEMBL3407433 0.82 ADORA2A (0.33) ALDH1A1MAPTHPGDMEN1GAA
SCHEMBL3090523 0.82 MAPT (0.49) ALDH1A1MAPTHPGDMEN1GAA
SCHEMBL3656837 0.80 ALDH1A1 (0.40) ALDH1A1MAPTHPGDMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197886-A1 5-CYANO-THIENOPYRIDINES FOR THE TREATMENT OF TUMORS Merck Patent GmbH (DE) 2010-06-23 EP claimed
WO-2009049743-A1 5-CYANO-THIENOPYRIDINES FOR THE TREATMENT OF TUMORS MERCK PATENT GMBH (DE) 2009-04-23 WO claimed