SCHEMBL3656355

SCHEMBL3656355

COc1ccc([N+](=O)[O-])c(CCNC2CCN(OC(=O)OC(C)(C)C)CC2C)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.39
RECQL P46063 2/20 0.39
LMNA P02545 3/20 0.39
MAPT P10636 5/20 0.36
MTNR1A P48039 3/20 0.36
MTNR1B P49286 3/20 0.36
PTPN1 P18031 1/20 0.35
MAPK1 P28482 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
HPGD P15428 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15752225 0.92 ALDH1A1 (0.36) ALDH1A1RECQLLMNAMAPTMTNR1A
SCHEMBL6525187 0.86 EPHX2 (0.43) ALDH1A1RECQLLMNAMAPTEPHX2
SCHEMBL3657873 0.86 EPHX2 (0.35) ALDH1A1MAPTMTNR1AHPGDSMN1; SMN2
SCHEMBL6525624 0.80 EPHX2 (0.44) ALDH1A1RECQLLMNAMAPTMAPK1
SCHEMBL3656515 0.78 EPHX2 (0.36) ALDH1A1RECQLLMNAMAPTMTNR1A
SCHEMBL6681269 0.73 PTPN1 (0.51) ALDH1A1LMNAMAPTMTNR1AMTNR1B
SCHEMBL6517994 0.72 EPHX2 (0.46) ALDH1A1MAPTMEN1KMT2AEPHX2
SCHEMBL30178371 0.72 ALDH1A1 (0.46) ALDH1A1RECQLLMNAMAPTMTNR1A
SCHEMBL28638738 0.72 ALDH1A1 (0.46) ALDH1A1RECQLLMNAMAPTMTNR1A
SCHEMBL17870715 0.72 ALDH1A1 (0.44) ALDH1A1RECQLLMNAMAPTPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205590-B1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-06-04 EP disclosed
EP-2205590-A1 CGRP ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-07-14 EP disclosed
WO-2009050232-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed