SCHEMBL3657412

SCHEMBL3657412

CN1CC2CCN(c3cncc(Br)c3)C2C1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 16/20 0.65
CHRNB2 P17787 4/20 0.51
CHRNA4 P43681 4/20 0.51
CHRNB4 P30926 3/20 0.51
CHRNA3 P32297 3/20 0.51
KCNH2 Q12809 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4113424 1.00 HRH3 (0.65) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4108977 0.88 CHRNB2 (0.61) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4920608 0.79 HRH3 (1.00) HRH3KCNH2
SCHEMBL4920616 0.79 HRH3 (1.00) HRH3KCNH2
SCHEMBL2410032 0.79 HRH3 (1.00) HRH3KCNH2
SCHEMBL2412379 0.75 HRH3 (1.00) HRH3KCNH2
SCHEMBL4113397 0.75 GPR119 (0.47) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4113401 0.75 GPR119 (0.47) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL3062935 0.74 HRH3 (0.60) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL24528539 0.73 CHRNB2 (0.49) CHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231672-A1 BIARYL SUBSTITUTED DIAZABICYCLOALKANE DERIVATIVES Abbott Laboratories (US) 2010-09-29 EP disclosed
WO-2009067586-A1 BIARYL SUBSTITUTED DIAZABICYCLOALKANE DERIVATIVES ABBOTT LABORATORIES (US) 2009-05-28 WO disclosed