SCHEMBL365767

SCHEMBL365767

CS(=O)(=O)NC(=O)c1ccc(OCc2ccccc2C(F)(F)F)cc1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.67
MAOA P21397 1/20 0.67
MMP13 P45452 3/20 0.53
ADAMTS4 O75173 2/20 0.53
SPHK2 Q9NRA0 4/20 0.52
SPHK1 Q9NYA1 4/20 0.52
SCN3A Q9NY46 1/20 0.49
ADAM17 P78536 3/20 0.48
MMP1 P03956 2/20 0.48
SRD5A2 P31213 1/20 0.46
PTPN1 P18031 1/20 0.46
MCL1 Q07820 1/20 0.45
SCN9A Q15858 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365141 0.84 MAOB (0.65) MAOBMMP13SCN3AADAM17MMP1
SCHEMBL16239897 0.82 MRGPRX4 (0.62) MAOBMAOASCN9AMRGPRX4
SCHEMBL364245 0.81 MAOA (0.65) MAOBMAOASCN3AADAM17MMP1
SCHEMBL2088377 0.81 MAOB (1.00) MAOBMAOAMMP13ADAMTS4SPHK2
SCHEMBL365920 0.81 RORC (0.62) SPHK2SPHK1SCN3AADAM17MMP1
SCHEMBL365343 0.80 MAOB (0.52) MAOBSCN3AMMP1MCL1SCN9A
SCHEMBL364125 0.80 FFAR1 (0.54) SCN3AADAM17PTPN1MCL1SCN9A
SCHEMBL365173 0.78 MAOB (0.61) MAOBSCN3ASRD5A2MCL1
SCHEMBL14890492 0.77 MAOA (0.52) MAOBMAOAMMP13ADAMTS4SCN3A
SCHEMBL363886 0.77 MAOB (0.69) MAOBMMP13ADAMTS4SPHK2SPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
EP-2593428-A2 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS Pfizer Limited (GB) 2013-05-22 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A MAOB 3660/4885MAOA 3705/4885MMP13 4508/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.